sales@targetmol.com (US) / info@targetmol.com    Tel: (781) 999-4286 / (781) 999-5354
Home > GPCR/G Protein > OX Receptor > SB408124

SB408124

Catalog No. T6658    CAS 288150-92-5    Synonyms: SB-408124

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

Pack Size Availability Price/USD Quantity
5 mg In Stock 50.00
10 mg In Stock 90.00
25 mg In Stock 162.00
50 mg In Stock 323.00
100 mg In Stock 582.00
1 mL * 10 mM (in DMSO) In Stock 51.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

Receptor:

OX1 (membrane); OX1 (whole cell);

Chemical Information:
Molecular Weight 356.37
Formula C19H18F2N4O
CAS Number 288150-92-5
Solubility

DMSO: 35.6 mg/mL (100 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Reference
Product Recommendations