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ZAP-180013

Catalog No. T8697 CAS 873080-25-2

ZAP-180013 is an inhibitor of zeta-chain-associated protein kinase 70 (ZAP70,IC50 : 1.8 μM).

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ZAP-180013, CAS 873080-25-2

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	ZAP-180013 is an inhibitor of zeta-chain-associated protein kinase 70 (ZAP70,IC50 : 1.8 μM).
Targets&IC50	ZAP-70:1.8 μM (IC50)

Molecular Weight	454.32
Formula	C19H17Cl2N3O4S
CAS No.	873080-25-2

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 250 mg/mL (550.26 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Patrick R Visperas, et al. Identification of Inhibitors of the Association of ZAP-70 With the T Cell Receptor by High-Throughput Screen. SLAS Discov. 2017 Mar;22(3):324-331.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Compound Library Inhibitor Library Immunology/Inflammation Compound Library Kinase Inhibitor Library Anti-Aging Compound Library Bioactive Compound Library Tyrosine Kinase Inhibitor Library

Related Products

Related compounds with same targets

Taxoquinone Isoderrone Buddlenoid A 3'-Deoxy-4-O-methylsappanol Viscumneoside III Trametenolic acid Kanzonol C Glabrene

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

ZAP-180013 873080-25-2 蛋白酪氨酸激酶蛋白酶体 Tyrosinase Tyrosine Kinases Inhibitor autoimmune ZAP-70 tyrosine T-cell ZAP 180013 ZAP180013 antigen inhibit inhibitor

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