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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6720 | Vatalanib dihydrochloride | CGP-797870 dihydrochloride , ZK-222584 dihydrochloride , Vatalanib 2HCl , PTK787 dihydrochloride , Vatalanib (PTK787) 2HCl , CGP-79787 dihydrochloride | VEGFR , Apoptosis , PDGFR |
Vatalanib dihydrochloride (PTK787 dihydrochloride)(IC50=37 nM) is an inhibitor of VEGFR2/KDR. It exhibits less effective against VEGFR1/Flt-1 and 18-fold against VEGFR3/Flt-4. |