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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T23515 | VU-29 | VU 29 | GluR |
VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes (EC50: rmGluR1/rmGluR2=557 nM/1.5 μM; hmGluR4=154 nM). |