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Metabolism PPAR VCE-004.8

VCE-004.8

Catalog No. T13289   CAS 1818428-24-8
Synonyms: VCE-​004.8,

VCE-004.8 is a specific dual agonist of PPARγ and CB2 receptor with potent anti-inflammatory activity. VCE-004.8 attenuates adipogenesis and prevents diet-induced obesity.

VCE-004.8, CAS 1818428-24-8
Pack Size Availability Price/USD Quantity
1 mg In stock 141.00
5 mg In stock 285.00
10 mg In stock 530.00
25 mg In stock 1010.00
1 mL * 10 mM (in DMSO) In stock 332.00
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Purity 99.22%
Biological Description
Chemical Properties
Storage & Solubility Information
Description VCE-004.8 is a specific dual agonist of PPARγ and CB2 receptor with potent anti-inflammatory activity. VCE-004.8 attenuates adipogenesis and prevents diet-induced obesity.
Targets&IC50 PPARγ
Synonyms VCE-​004.8 ,
Purity 99.22%
Molecular Weight 433.58
Formula C28H35NO3
CAS No. 1818428-24-8

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

DMSO: 49 mg/mL (113.01 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Navarrete C, et al. Hypoxia mimetic activity of VCE-004.8, a cannabidiol quinone derivative: implications for multiple sclerosis therapy. J Neuroinflammation. 2018 Mar 1;15(1):64. 2. Palomares B, et al. VCE-004.8, A Multitarget Cannabinoquinone, Attenuates Adipogenesis and Prevents Diet-Induced Obesity. Sci Rep. 2018 Oct 31;8(1):16092.

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