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P276-00

Catalog No. T6924    CAS 920113-03-7   

P276-00 is a novel CDK1, CDK4 and CDK9 inhibitor with IC50 of 79 nM, 63 nM and 20 nM, respectively. Phase 2/3.

Pack Size Availability Price/USD Quantity
1 mg Inquiry 62.00
2 mg Inquiry 111.00
5 mg Inquiry 200.00
10 mg Inquiry 320.00
25 mg Inquiry 576.00
1 mL * 10 mM (in DMSO) Inquiry 200.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

P276-00 is a novel CDK1, CDK4 and CDK9 inhibitor with IC50 of 79 nM, 63 nM and 20 nM, respectively. Phase 2/3.

Receptor:

CDK1/CyclinB; CDK2/CyclinA; CDK4/CyclinD1; CDK6/CyclinD3; CDK9/CyclinT1;

Chemical Information:
Molecular Weight 438.30
Formula C21H20ClNO5·HCl
CAS Number 920113-03-7
Solubility

DMSO: 82 mg/mL (187.1 mM)

Ethanol: 7 mg/mL (15.97 mM)

Water: 81 mg/mL (184.8 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Reference
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