Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant. |
In vitro | For antagonistic activity, (?)-mavoglurant, the (?)-enantiomer shows IC50 of 0.11 μM and 0.03 μM (Ca2+ and PI-turnover) whereas the (+)-enantiomer ((+)-10) shows only 37% and 18% inhibition at 10 μM. |
Synonyms | AFQ-056 racemate |
Molecular Weight | 313.39 |
Formula | C19H23NO3 |
CAS No. | 1636881-61-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (159.55 mM), sonification is recommended.
You can also refer to dose conversion for different animals. More
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Mavoglurant racemate 1636881-61-2 Others AFQ-056 racemate inhibitor inhibit