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Metabolism PPAR INT-131

INT-131

Catalog No. T8780   CAS 315224-26-1
Synonyms: CHS 131, AMG-131,

INT-131, is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, which can be used for the treatment of type 2 diabetes mellitus (non-insulin dependent diabetes)

INT-131, CAS 315224-26-1
Pack Size Availability Price/USD Quantity
1 mg In stock 131.00
5 mg In stock 368.00
10 mg In stock 551.00
25 mg In stock 1102.00
50 mg In stock 1433.00
100 mg In stock 1862.00
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Biological Description
Chemical Properties
Storage & Solubility Information
Description INT-131, is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, which can be used for the treatment of type 2 diabetes mellitus (non-insulin dependent diabetes)
Targets&IC50
Synonyms CHS 131 , AMG-131 ,
Purity 98.01%
Molecular Weight 514.21
Formula C21H12Cl4N2O3S
CAS No. 315224-26-1

Storage

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Kintscher U , Goebel M . INT-131, a PPARgamma agonist for the treatment of type 2 diabetes.[J]. Curr Opin Investig Drugs, 2009, 10(4):381-387.

Related Products

Related compounds with same targets
INT-131 12-O-Methylcarnosic acid Oleoylethanolamide GW1929 GW 6471 3-Guanidinopropionic Acid Growth hormone releasing peptide Ailanthoidol

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