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GSK690693

Catalog No. T6285    CAS 937174-76-0   

GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.

Pack Size Availability Price/USD Quantity
2 mg In stock 51.00
5 mg In stock 80.00
10 mg In stock 125.00
25 mg In stock 226.00
100 mg In stock 720.00
1 mL * 10 mM (in DMSO) In Stock 91.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.

Receptor:

Akt1; Akt3; PKCη; PKCθ; PrkX;

Chemical Information:
Molecular Weight 425.48
Formula C21H27N7O3
CAS Number 937174-76-0
Solubility

DMSO: 21.3 mg/mL (50 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.