Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe. The pIC50 of GSK4028 is 4.9 in a TR-FRET assay.
Description | GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe. The pIC50 of GSK4028 is 4.9 in a TR-FRET assay. |
Targets&IC50 | PCAF/GCN5:4.9(pIC50) |
In vitro | GSK4028 also demonstrates potency toward BRD4 BD1 and BRD9 inTR-FRET assay with pIC50s of <4.3 and 4.5±0.13, respectively.GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9. |
Molecular Weight | 377.28 |
Formula | C17H21BrN4O |
CAS No. | 2079886-19-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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GSK4028 2079886-19-2 Others GSK-4028 GSK 4028 inhibitor inhibit