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Fasudil hydrochloride

Catalog No. T3060    CAS 105628-07-7    Synonyms: AT-877, Fasudil HCl, HA-1077, Fasudil (HA-1077) HCl, HA-1077 hydrochloride

Fasudil Hydrochloride is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.

Pack Size Availability Price/USD Quantity
100 mg In stock 51.00
200 mg In stock 78.00
500 mg In stock 131.00
1 mL * 10 mM (in DMSO) In stock 50.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

Fasudil Hydrochloride is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.

Receptor:

MLCK; PKA; PKC; PKG; ROCK2;

Chemical Information:
Molecular Weight 327.83
Formula C14H18ClN3O2S
CAS Number 105628-07-7
Solubility

DMSO: 24.6 mg/mL (75 mM)

water: 32.8 mg/mL (100 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.