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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T19913 | CKI-7 | CKI 7 2HCl , CKI-7 dihydrochloride , CKI7 2HCl , CKI 7 dihydrochloride , CKI7 dihydrochloride , CKI-7 2HCl | CDK , S6 Kinase , Casein Kinase , SGK , ROCK |
CKI-7 is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor. CKI-7 also inhibits SGK, ribosomal S6 kinase-1 (S6K1), and MSK1. |