Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 34.00 | |
2 mg | In stock | $ 48.00 | |
5 mg | In stock | $ 79.00 | |
10 mg | In stock | $ 143.00 | |
25 mg | In stock | $ 279.00 | |
50 mg | In stock | $ 485.00 | |
100 mg | In stock | $ 715.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 88.00 |
Description | CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM). |
Targets&IC50 | GABAB:85 nM |
Kinase Assay | Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000). |
Synonyms | CGP 52432 |
Molecular Weight | 384.24 |
Formula | C15H24Cl2NO4P |
CAS No. | 139667-74-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5 mg/mL (13.01 mM), Sonication and heating are recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
CGP52432 139667-74-6 Membrane transporter/Ion channel Neuroscience GABA Receptor Inhibitor inhibit Gamma-aminobutyric acid Receptor CGP 52432 γ-Aminobutyric acid Receptor CGP-52432 inhibitor