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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7709 | (E/Z)-GSK5182 | GSK5182(Z/E) | Estrogen/progestogen Receptor , ROS |
(E/Z)-GSK5182 (GSK5182(Z/E)) is a racemic mixture comprising (E)-GSK5182 and (Z)-GSK5182 isomers. It acts as a highly selective and orally active inverse agonist for the estrogen-related receptor γ (ERRγ), demonstrating ... | |||
T8370 | GSK5182 | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Reactive Oxygen Species | |
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM) |