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Kinase Inhibitor Library

Catalog No. L1600

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. Aprotein kinasemodifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved insignal transduction. Various other kinases act on small molecules such aslipids,carbohydrates,amino acids, andnucleotides, either for signaling or to prime them for metabolic pathways.

TargetMol’s Tyrosine Kinase Inhibitors Library, containing 860 kinase inhibitors, can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

Pack Size	Price
100 μL * 10 mM (in DMSO)	USD 12025.00
250 μL * 10 mM (in DMSO)	USD 19670.00
1 mg	USD 19670.00

Product Description

A unique collection of 860 GPCR-active agents for high throughput screening and high content screening for GPCR drug discovery, and new GPCR target identification and research;
Potential to find new GPCR drug candidates by screening against orphan GPCRs;
Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
Targets include 5-HT receptor, dopamine receptor, opioid receptor, adrenergic receptor, mGluR, Cannabinoid receptor, ETA-receptor, etc;
Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
Structurally diverse, medicinally active, and cell permeable;
NMR and HPLC validated to ensure high purity and quality;

The compound library can be highly customized. You can select compounds, quantities, format (dry/solid or DMSO), plate map, and concentration to meet your specific requirement. Please check our Compound Library Instructions for more information.

Packaging and Storage

Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
Shipped with blue ice; Stable for One year as powder, 6 months at - 20 ° C in DMSO or 12months at -80 ° C in DMSO

Library Composition

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