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Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones Enzyme GPCR/G Protein Immunology / Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology&virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries Approved / Repurposing Characteristic Bioactive Libraries COVID-19 / SARS-CoV-2 Disease Focused Target / Pathway Focused Natural Product Libraries Characteristic Natural Product Libraries Natural Compound Library for HTS Fragment Libraries Diversity Sets Custom Compound Library
Signaling pathway Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones Enzyme GPCR/G Protein Immunology / Inflammation JAK/STAT signaling MAPK
Membrane transporter/Ion channel Metabolism Microbiology&virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling
Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Focused Bioactive Libraries Approved / Repurposing Characteristic Bioactive Libraries COVID-19 / SARS-CoV-2 Disease Focused Target / Pathway Focused
Natural Product Libraries Characteristic Natural Product Libraries Natural Compound Library for HTS Diversity Sets Golden Scaffold Library Mini Scaffold Library
Fragment Libraries Drug-fragment Library Featured Fragment Library High Solubility Fragment Library Custom Compound Library
Compound Libraries Inhibitor Library

Inhibitor Library

Catalog No. L2000
  Library Compound List   Excel SDF

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 3809 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 32920.00
250 μL * 10 mM (in DMSO) 54910.00
1 mg 54910.00
Top Publication Citing Use of Targetmol Products
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Product Description

  • A unique collection of 3809 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging and Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice.

Supporting Files

Library Handling Instructions (927 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2000)

Library Composition

AChR (128)
5-HT Receptor (124)
Adrenergic Receptor (99)
COX (99)
Dopamine Receptor (77)
DNA/RNA Synthesis (72)
Histamine Receptor (67)
EGFR (64)
PI3K (61)
VEGFR (59)
Estrogen/progestogen Receptor (56)
Sodium Channel (53)
CDK (50)
Potassium Channel (49)
Topoisomerase (44)
Dehydrogenase (43)
Calcium Channel (42)
Src (42)
PDGFR (41)
HDAC (41)
Bcr-Abl (39)
Antibacterial (38)
GR (37)
FLT (37)
GABA Receptor (36)
PDE (36)
JAK (36)
mTOR (35)
PPAR (34)
P450 (33)
FGFR (33)
c-Kit (33)
Microtubule Associated (32)
NF-κB (31)
RAAS (31)
ribosome (30)
Autophagy (30)
Vitamin (29)
ALK (28)
Epigenetic Reader Domain (27)
Raf (27)
PKC (27)
GluR (26)
Histone Methyltransferase (26)
GSK-3 (25)
c-Met/HGFR (25)
Androgen Receptor (24)
HIV Protease (24)
Antibiotic (23)
MAO (23)
Amino Acids and Derivatives (22)
Carbonic Anhydrase (20)
Norepinephrine (20)
p38 MAPK (20)
Tyrosine Kinases (19)
Antifection (19)
ATPase (19)
Aurora Kinase (19)
Akt (18)
GPR (18)
DNA-PK (18)
TNF (18)
MEK (18)
MRP (16)
NMDAR (16)
ERK (16)
IL Receptor (16)
IGF-1R (15)
IκB/IKK (15)
Wnt/beta-catenin (15)
Proteasome (14)
ROS (14)
Reverse Transcriptase (14)
MMP (14)
DNA Alkylation (14)
ATM/ATR (14)
HSP (13)
Opioid Receptor (13)
Serine Protease (13)
PKA (13)
TRP/TRPV Channel (13)
STAT (13)
TGF-beta/Smad (13)
TAM Receptor (12)
Trk receptor (12)
Prostaglandin Receptor (12)
Retinoid Receptor (12)
PARP (12)
Phospholipase (12)
p53 (12)
HER (12)
FAK (12)
c-RET (12)
Cysteine Protease (12)
Chk (11)
Caspase (11)
Adenosine Receptor (11)
HIF (11)
Hedgehog/Smoothened (11)
NADPH (11)
ROCK (11)
S6 Kinase (11)
Transferase (11)
Thrombin (11)
Sirtuin (10)
PLK (10)
Mdm2 (10)
JNK (10)
P2 Receptor (10)
Gamma-secretase (10)
DNA gyrase (10)
DHFR (10)
DPP-4 (10)
BTK (10)
CaMK (10)
CFTR (10)
BCL (9)
Casein Kinase (9)
CAT (9)
HMG-CoA Reductase (9)
NOS (9)
Proton pump (9)
Serine/threonin kinase (9)
Tyrosinase (9)
Syk (8)
Thyroid hormone receptor(THR) (8)
S1P Receptor (8)
PDK (8)
Lipoxygenase (8)
LRRK2 (8)
Histone Demethylase (8)
DUB (8)
Glucokinase (8)
Cannabinoid Receptor (8)
AMPK (8)
CCR (7)
CXCR (7)
ABC (7)
AhR (7)
Aromatase (7)
Antifungal (7)
FXR (7)
HCV Protease (7)
MAPK (7)
SGLT (7)
Sigma receptor (6)
Reductase (6)
Lipid (6)
Kinesin (6)
Integrin (6)
NOD (6)
HSV (6)
IAP (6)
Glucocorticoid Receptor (6)
FAAH (6)
Factor Xa (6)
DNA Methyltransferase (6)
Antioxidant (6)
Antiviral (6)
Apoptosis inducer (6)
Annexin A (6)
Beta Amyloid (6)
CSF-1R (5)
c-Fms (5)
Endothelin Receptor (5)
Fatty Acid Synthase (5)
MPO (5)
Nucleoside Antimetabolite/Analog (5)
OX Receptor (5)
Pim (5)
Phosphatase (5)
LTR (5)
Rho (5)
TLR (5)
UGT (5)
Vasopressin Receptor (4)
transporter (4)
Telomerase (4)
PYK2 (4)
Lipase (4)
Liver X Receptor (4)
Monocarboxylate transporter (4)
OCT (4)
p97 (4)
IDO (4)
Hydroxylase (4)
Influenza Virus (4)
HIF/HIF Prolyl-Hydroxylase (4)
HBV (4)
Cell wall (4)
CETP (4)
Arginase (4)
BACE (3)
advanced glycation end products (3)
ACAT (3)
Chloride channel (3)
cholecystokinin (3)
CRM1 (3)
c-Myc (3)
Glutathione reductase (3)
Ferroptosis (3)
Free radical scavengers (3)
GluCls (3)
Dynamin (3)
DYRK (3)
Neurokinin 1 (3)
P-gp (3)
PERK (3)
MTH1 (3)
Na-K-Cl cotransporter (3)
LDL (3)
Porcupine (3)
Protease-activated Receptor (3)
Platelet aggregation (3)
SGK (3)
Somatostatin (2)
ROR (2)
PTEN (2)
Ras (2)
Tie-2 (2)
KSP (2)
lysosomal autophagy (2)
NADPH-oxidase (2)
MLK (2)
PGE Synthase (2)
Phosphorylase (2)
PD-1/PD-L1 (2)
PAFR (2)
Nrf2 (2)
Ephrin Receptor (2)
DNA (2)
Gap Junction Protein (2)
Hck (2)
GPCR19 (2)
GST (2)
Decarboxylase (2)
BMI-1 (2)
cAMP (2)
Acetyl-CoA Carboxylase (2)
ACK (2)
ASK (2)
ATP Citrate Lyase (2)
Adiponectin receptor (1)
Aminopeptidase (1)
Bombesin Receptor (1)
CaSR (1)
cell cycle arrest (1)
GTPase (1)
GSNOR (1)
GlyT (1)
GNRH Receptor (1)
GPX (1)
GRK (1)
Integrase (1)
Hydrogenase (1)
Glucagon Receptor (1)
FOXO1 (1)
DprE1 (1)
E1/E2/E3 Enzyme (1)
PAI-1 (1)
OAT (1)
NPC1L1 (1)
PED (1)
Monoamine Transporter (1)
Melatonin Receptor (1)
MELK (1)
NAMPT (1)
MALT (1)
LPA Receptor (1)
LHRH (1)
Thioredoxin (1)
Survivin (1)
VDA (1)
Wee1 (1)
RAR/RXR (1)
PKM (1)
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