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Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Inhibitor Library

Catalog No. L2000
  Library Compound List   Excel SDF

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 7618 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
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Product Description

  • A unique collection of 7618 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2000)

Library Composition

Apoptosis (762)
Autophagy (583)
Antibacterial (436)
Antibiotic (252)
5-HT Receptor (214)
Endogenous Metabolite (200)
COX (192)
CDK (176)
DNA/RNA Synthesis (167)
NF-κB (160)
HIV Protease (159)
PI3K (159)
AChR (156)
EGFR (149)
Dopamine Receptor (143)
VEGFR (141)
Parasite (129)
Antifungal (128)
Adrenergic Receptor (127)
Epigenetic Reader Domain (125)
P450 (121)
PDE (120)
Dehydrogenase (120)
Histamine Receptor (118)
Histone Methyltransferase (107)
HDAC (106)
Potassium Channel (103)
Calcium Channel (96)
JAK (91)
FLT (89)
Src (88)
PDGFR (87)
mTOR (87)
Influenza Virus (86)
Sodium Channel (82)
Topoisomerase (82)
Microtubule Associated (80)
Phosphatase (78)
SARS-CoV (75)
FGFR (74)
Akt (73)
ERK (73)
STAT (72)
TRP/TRPV Channel (72)
AChE (71)
Reactive Oxygen Species (70)
Raf (69)
c-Kit (67)
PKC (67)
p38 MAPK (66)
PARP (66)
TNF (65)
Wnt/beta-catenin (62)
c-Met/HGFR (62)
HCV Protease (61)
Prostaglandin Receptor (59)
RAAS (58)
Bcr-Abl (58)
Ferroptosis (58)
Proteasome (57)
GABA Receptor (57)
Ras (56)
BCL (53)
GSK-3 (53)
Aurora Kinase (52)
MMP (52)
Virus Protease (50)
ALK (50)
Lipoxygenase (49)
MAO (49)
PPAR (47)
Adenosine Receptor (46)
HSP (46)
NMDAR (46)
Phospholipase (45)
NO Synthase (45)
Tyrosinase (44)
IL Receptor (43)
Antioxidant (43)
TGF-beta/Smad (42)
MEK (41)
iGluR (41)
JNK (41)
DUB (41)
E1/E2/E3 Enzyme (41)
Beta Amyloid (41)
GluR (40)
ATPase (39)
Mitophagy (39)
Tyrosine Kinases (39)
Monoamine Oxidase (39)
BTK (38)
GPR (38)
CCR (38)
Caspase (38)
Casein Kinase (38)
HER (37)
DNA-PK (37)
Reverse Transcriptase (37)
HSV (36)
P-gp (36)
Serine/threonin kinase (36)
ROCK (36)
MAPK (36)
HBV (35)
IκB/IKK (35)
Histone Demethylase (35)
CXCR (34)
Sirtuin (34)
AMPK (34)
HIF/HIF Prolyl-Hydroxylase (34)
Androgen Receptor (34)
Serotonin Transporter (34)
Transferase (33)
Interleukin (33)
Mitochondrial Metabolism (33)
Estrogen Receptor/ERR (33)
Cysteine Protease (33)
Estrogen/progestogen Receptor (33)
c-RET (32)
CaMK (32)
Nucleoside Antimetabolite/Analog (32)
TAM Receptor (32)
Integrin (32)
HIF (31)
TLR (31)
PKA (31)
Anti-infection (30)
NOS (29)
ROS (29)
Serine Protease (28)
Gamma-secretase (28)
Carbonic Anhydrase (28)
S6 Kinase (27)
Trk receptor (27)
Histone Acetyltransferase (27)
IGF-1R (27)
Proton pump (27)
Drug Metabolite (27)
Opioid Receptor (27)
P2X Receptor (26)
Norepinephrine (26)
Hedgehog/Smoothened (25)
FAK (25)
FAAH (25)
PLK (25)
c-Fms (24)
Reductase (24)
RIP kinase (24)
DPP-4 (23)
Glucosidase (23)
Indoleamine 2,3-Dioxygenase (IDO) (23)
DNA Methyltransferase (23)
Cannabinoid Receptor (23)
ribosome (22)
Syk (22)
Glucocorticoid Receptor (22)
Fatty Acid Synthase (21)
Antiviral (21)
p53 (21)
Kinesin (20)
Neurokinin receptor (20)
Pim (20)
Chk (20)
ATM/ATR (20)
SGLT (19)
Antifection (19)
HMG-CoA Reductase (19)
Nrf2 (19)
LPL Receptor (19)
S1P Receptor (18)
Chloride channel (18)
LRRK2 (18)
transporter (17)
Lipase (17)
Complement System (17)
Acyltransferase (17)
NOD (17)
Mdm2 (17)
Smo (17)
PAK (17)
Endothelin Receptor (17)
PDK (17)
OX Receptor (16)
Leukotriene Receptor (16)
Epoxide Hydrolase (16)
NADPH (16)
MRP (16)
IRAK (15)
NOD-like Receptor (NLR) (15)
P2Y Receptor (15)
Xanthine Oxidase (15)
Rho (15)
Glutathione Peroxidase (15)
BACE (14)
IRE1 (14)
Hydroxylase (14)
DYRK (14)
c-Myc (14)
Thrombin (13)
Retinoid Receptor (13)
CSF-1R (13)
Sigma receptor (13)
cAMP (13)
LTR (13)
Glucokinase (13)
PI4K (13)
PGE Synthase (13)
Aryl Hydrocarbon Receptor (12)
LPA Receptor (12)
PD-1/PD-L1 (12)
Ephrin Receptor (12)
Immunology/Inflammation related (12)
Aminopeptidase (12)
Antifolate (12)
PERK (12)
Protease-activated Receptor (12)
Acetyl-CoA Carboxylase (11)
AhR (11)
IDO (11)
Aromatase (11)
Neuropeptide Y Receptor (11)
Beta-Secretase (11)
Stearoyl-CoA Desaturase (SCD) (11)
Isocitrate Dehydrogenase (IDH) (11)
Factor Xa (11)
ROS Kinase (11)
STING (11)
GTPase (10)
Myosin (10)
DHFR (10)
PAI-1 (10)
Discoidin Domain Receptor (DDR) (10)
Vasopressin Receptor (10)
Melanocortin Receptor (9)
GNRH Receptor (9)
IAP (9)
SGK (9)
ATP Citrate Lyase (9)
Monoamine Transporter (9)
Telomerase (9)
RSV (9)
cholecystokinin (9)
Monocarboxylate transporter (9)
NAMPT (8)
CETP (8)
DNA gyrase (8)
YAP (8)
BCRP (8)
Porcupine (8)
PAD (8)
Phosphorylase (8)
NADPH-oxidase (7)
PTEN (7)
p97 (7)
ROR (7)
Na+/Ca2+ Exchanger (7)
Neprilysin (7)
GRK (7)
Lipid (7)
CFTR (7)
Tie-2 (7)
DNA (7)
ASK (7)
Ligands for Target Protein for PROTAC (7)
MLK (6)
MNK (6)
Guanylate cyclase (6)
Dynamin (6)
Adenylyl cyclase (6)
MAGL (6)
OAT (6)
SIK (6)
Platelet aggregation (6)
ABC (6)
TOPK (5)
Adenosine deaminase (5)
CAT (5)
APC (5)
Aquaporin (5)
Neurotensin Receptor (5)
BMI-1 (5)
Bradykinin Receptor (5)
Thyroid hormone receptor(THR) (5)
LIM Kinase (5)
GlyT (5)
Liver X Receptor (5)
GPX (5)
PAFR (5)
CRFR (5)
Carboxypeptidase (5)
cGAS (5)
CRISPR/Cas9 (5)
FLAP (5)
Wee1 (5)
CRM1 (5)
Progesterone Receptor (5)
MELK (5)
MTH1 (5)
DprE1 (5)
Glutaminase (5)
Gap Junction Protein (5)
UGT (5)
DNA Alkylator/Crosslinker (5)
Glucagon Receptor (5)
GST (5)
Arginase (4)
VDAC (4)
PYK2 (4)
IFNAR (4)
ACK (4)
CaSR (4)
Decarboxylase (4)
NPC1L1 (4)
Hck (4)
MALT (4)
Amino Acids and Derivatives (4)
Methionine Adenosyltransferase (MAT) (4)
DNA Alkylation (4)
Ligand for E3 Ligase (4)
LDL (4)
Bombesin Receptor (4)
Survivin (4)
Angiotensin-converting Enzyme (ACE) (4)
CGRP Receptor (4)
NEDD8 (4)
Galectin (4)
MT Receptor (4)
KSP (4)
CD73 (3)
PKM (3)
AAK1 (AP2 associated kinase 1) (3)
Hexokinase (3)
Melatonin Receptor (3)
MyD88 (3)
CD38 (3)
Hippo pathway (3)
Pyroptosis (3)
OXPHOS (3)
Imidazoline Receptor (3)
FXR (3)
RANKL/RANK (2)
RAR/RXR  (2)
hCE (2)
GHSR (2)
Na-K-Cl cotransporter (2)
Transaminase (2)
KLF (2)
Integrase (2)
Prolyl Endopeptidase (PREP) (2)
Melanin-concentrating Hormone Receptor (MCHR) (2)
TSH Receptor (2)
Necroptosis (2)
advanced glycation end products (2)
Apelin receptor (2)
Fas/FasL (2)
EBI2/GPR183 (2)
Somatostatin (2)
LHRH (2)
Oxytocin Receptor (2)
Haspin Kinase (2)
Free radical scavengers (2)
HCN Channel (2)
PROTACs (1)
PROTAC Linker (1)
Protease (1)
Cell wall (1)
Fer/FerT kinase (1)
gp120/CD4 (1)
lysosomal autophagy (1)
Neuropeptide W (1)
Taste receptor (1)
Stemness kinase (1)
GPCR19 (1)
Thioredoxin (1)
stilbene oxidase (1)
Anion Exchanger (1)
VDA (1)
cell cycle arrest (1)
PGC-1α (1)
N-Acetylglucosaminyltransferase (1)
DAPK (1)
aconitase (1)
GSNOR (1)
NUDIX hydrolase (1)
GluCls (1)
FABP (1)
Molecular Glues (1)
Annexin A (1)
FOXO1 (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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