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Compound Libraries FDA-approved Drug Library

FDA-approved Drug Library

Catalog No. L4200
  Library Compound List   Excel SDF

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 7180.00
250 μL * 10 mM (in DMSO) 14114.00
1 mg 14114.00
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Product Description

  • A unique collection of 1436 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L4200)

Library Composition

Adrenergic Receptor (83)
AChR (78)
5-HT Receptor (74)
Antibiotic (50)
Dopamine Receptor (50)
Histamine Receptor (47)
COX (46)
Antibacterial (45)
DNA/RNA Synthesis (44)
Potassium Channel (39)
Glucocorticoid Receptor (37)
Estrogen/progestogen Receptor (36)
Sodium Channel (36)
GR (32)
Topoisomerase (25)
Vitamin (22)
PDE (21)
Calcium Channel (21)
Autophagy (20)
ribosome (20)
RAAS (19)
Dehydrogenase (19)
GABA Receptor (19)
Norepinephrine (19)
Antifection (18)
VEGFR (18)
HIV Protease (17)
Microtubule Associated (15)
Carbonic Anhydrase (15)
Antifungal (13)
MRP (13)
HCV Protease (13)
Reverse Transcriptase (13)
PPAR (13)
P450 (12)
DNA Alkylation (12)
c-Kit (12)
EGFR (12)
PDGFR (11)
ROS (9)
DHFR (9)
ATPase (9)
MAO (9)
HDAC (8)
GluR (8)
Bcr-Abl (8)
Androgen Receptor (8)
Proton pump (8)
Tyrosine Kinases (8)
Src (8)
Retinoid Receptor (7)
TNF (7)
Raf (7)
ABC (7)
DNA gyrase (7)
FGFR (7)
NMDAR (7)
Opioid Receptor (7)
NADPH (7)
NF-κB (6)
HMG-CoA Reductase (6)
FLT (6)
Amino Acids and Derivatives (6)
Prostaglandin Receptor (6)
Thrombin (6)
Thyroid hormone receptor(THR) (5)
Transferase (5)
P2 Receptor (5)
Proteasome (5)
Annexin A (5)
CaMK (5)
Factor Xa (5)
Endogenous Metabolite (4)
DPP-4 (4)
DNA Methyltransferase (4)
CDK (4)
CAT (4)
ALK (4)
IL Receptor (4)
Neurokinin receptor (4)
NOS (4)
JAK (4)
Lipoxygenase (4)
HBV (4)
MMP (4)
SGLT (4)
Parasite (4)
PI3K (4)
PKC (3)
PARP (3)
Phosphatase (3)
Phospholipase (3)
Reductase (3)
TRP/TRPV Channel (3)
Tyrosinase (3)
TLR (3)
STAT (3)
MPO (3)
MT Receptor (3)
MEK (3)
mTOR (3)
Na-K-Cl cotransporter (3)
Influenza Virus (3)
Integrin (3)
GST (3)
Glutathione reductase (3)
Hedgehog/Smoothened (3)
AhR (3)
Arginase (3)
Aromatase (3)
CFTR (3)
Chloride channel (3)
Decarboxylase (3)
Endothelin Receptor (3)
Fatty Acid Synthase (3)
Free radical scavengers (2)
FXR (2)
BTK (2)
c-Met/HGFR (2)
Chk (2)
Cell wall (2)
c-RET (2)
BCL (2)
Adenosine Receptor (2)
Antiviral (2)
HER (2)
HIF (2)
GluCls (2)
GPR (2)
Glucokinase (2)
HSV (2)
IGF-1R (2)
Nucleoside Antimetabolite/Analog (2)
MAPK (2)
LDL (2)
Lipid (2)
Mitophagy (2)
TAM Receptor (2)
UGT (2)
Vasopressin Receptor (2)
Rho (2)
Phosphorylase (1)
Sigma receptor (1)
Sirtuin (1)
ROCK (1)
S1P Receptor (1)
S6 Kinase (1)
Serine Protease (1)
Serotonin Transporter (1)
PDK (1)
PED (1)
PKM (1)
Platelet aggregation (1)
PLK (1)
Protease-activated Receptor (1)
VDA (1)
Telomerase (1)
TGF-beta/Smad (1)
Syk (1)
Wnt/beta-catenin (1)
Monoamine Oxidase (1)
Monoamine Transporter (1)
MTH1 (1)
LTR (1)
lysosomal autophagy (1)
Melatonin Receptor (1)
OAT (1)
NPC1L1 (1)
Nrf2 (1)
Neprilysin (1)
NADPH-oxidase (1)
NKCC (1)
iGluR (1)
HSP (1)
IκB/IKK (1)
Integrase (1)
Hydrogenase (1)
Hydroxylase (1)
IAP (1)
Guanylate cyclase (1)
Histone Demethylase (1)
Histone Methyltransferase (1)
Gap Junction Protein (1)
GlyT (1)
GPCR19 (1)
GRK (1)
GSK-3 (1)
AMPK (1)
Akt (1)
AChE (1)
ACK (1)
ATM/ATR (1)
ATP Citrate Lyase (1)
CCR (1)
Caspase (1)
CaSR (1)
Beta-Secretase (1)
CXCR (1)
DNA Alkylator/Crosslinker (1)
CETP (1)
Ferroptosis (1)
Epigenetic Reader Domain (1)
Electron transport (1)
DUB (1)