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Compound Libraries FDA-approved Drug Library

FDA-approved Drug Library

Catalog No. L4200
  Library Compound List   Excel SDF

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

In addtion, we provide the peptides and other drug molecules with low solution stability in the form of dry powder (set as Part B) in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 8350.00
250 μL * 10 mM (in DMSO) 15448.00
1 mg 15448.00
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Product Description

  • A unique collection of 1470 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L4200)

Library Composition

Adrenergic Receptor (92)
AChR (88)
5-HT Receptor (82)
Antibacterial (56)
Dopamine Receptor (56)
Antibiotic (50)
Histamine Receptor (47)
COX (46)
DNA/RNA Synthesis (44)
Glucocorticoid Receptor (42)
Sodium Channel (42)
Estrogen/progestogen Receptor (41)
Potassium Channel (40)
GR (35)
HIV Protease (29)
Calcium Channel (27)
Topoisomerase (27)
Vitamin (25)
ribosome (25)
RAAS (24)
PDE (22)
GABA Receptor (22)
Autophagy (21)
VEGFR (20)
Dehydrogenase (19)
Antifection (18)
HCV Protease (18)
Norepinephrine (18)
Microtubule Associated (16)
EGFR (16)
Carbonic Anhydrase (16)
c-Kit (16)
Antifungal (15)
P450 (15)
PDGFR (14)
Reverse Transcriptase (13)
PPAR (13)
Androgen Receptor (13)
MRP (13)
MAO (12)
DNA Alkylation (12)
Endogenous Metabolite (11)
Prostaglandin Receptor (11)
Opioid Receptor (11)
Tyrosine Kinases (10)
DHFR (10)
Bcr-Abl (10)
FGFR (10)
GluR (9)
HDAC (9)
JAK (9)
ATPase (8)
ALK (8)
c-Met/HGFR (8)
c-RET (8)
CDK (8)
DNA gyrase (8)
Thrombin (8)
Src (8)
Raf (8)
Proton pump (7)
PI3K (7)
ROS (7)
Retinoid Receptor (7)
ABC (7)
HMG-CoA Reductase (7)
FLT (7)
NADPH (6)
MMP (6)
TAM Receptor (6)
Thyroid hormone receptor(THR) (6)
PARP (6)
NMDAR (6)
NF-κB (5)
Proteasome (5)
Transferase (5)
TNF (5)
SGLT (5)
IL Receptor (5)
Influenza Virus (5)
Lipoxygenase (5)
GNRH Receptor (5)
HER (5)
HBV (5)
Amino Acids and Derivatives (5)
Annexin A (5)
CaMK (5)
Aromatase (5)
Factor Xa (5)
DNA Methyltransferase (4)
DPP-4 (4)
CFTR (4)
Adenosine Receptor (4)
CAT (4)
GPR (4)
Hedgehog/Smoothened (4)
MEK (4)
MPO (4)
NOS (4)
mTOR (4)
STAT (4)
S1P Receptor (4)
Trk receptor (4)
TRP/TRPV Channel (4)
PKC (4)
P2 Receptor (4)
Phospholipase (4)
Reductase (3)
Tyrosinase (3)
TLR (3)
Vasopressin Receptor (3)
Serotonin Transporter (3)
Neurokinin receptor (3)
Na-K-Cl cotransporter (3)
MT Receptor (3)
Integrin (3)
GST (3)
Hydroxylase (3)
BTK (3)
BCL (3)
Antiviral (3)
AhR (3)
Fatty Acid Synthase (3)
Endothelin Receptor (3)
CaSR (2)
Chk (2)
Chloride channel (2)
Cell wall (2)
CXCR (2)
Cysteine Protease (2)
Decarboxylase (2)
AMPK (2)
AChE (2)
Arginase (2)
ATP Citrate Lyase (2)
Guanylate cyclase (2)
GPCR19 (2)
Glutathione reductase (2)
Free radical scavengers (2)
FXR (2)
LDL (2)
Lipid (2)
HSV (2)
MAPK (2)
Histone Methyltransferase (2)
Monoamine Oxidase (2)
Monoamine Transporter (2)
Neprilysin (2)
SARS-CoV (2)
ROCK (2)
Syk (2)
Sigma receptor (2)
UGT (2)
Wnt/beta-catenin (2)
Rho (2)
Protease-activated Receptor (2)
Parasite (2)
Nucleoside Antimetabolite/Analog (2)
OAT (1)
NKCC (1)
Phosphorylase (1)
PDK (1)
PED (1)
Phosphatase (1)
PKM (1)
Platelet aggregation (1)
PLK (1)
RAR/RXR (1)
VDA (1)
Thrombopoietin Receptor (1)
Sirtuin (1)
Somatostatin (1)
Telomerase (1)
TGF-beta/Smad (1)
ROR (1)
S6 Kinase (1)
Serine Protease (1)
NPC1L1 (1)
Nrf2 (1)
MTH1 (1)
NADPH-oxidase (1)
LTR (1)
lysosomal autophagy (1)
Melanocortin Receptor (1)
Melatonin Receptor (1)
Mitochondrial Metabolism (1)
Mitophagy (1)
Hydrogenase (1)
Integrase (1)
IκB/IKK (1)
Electron transport (1)
Gap Junction Protein (1)
GluCls (1)
GlyT (1)
Glucokinase (1)
GRK (1)
GSK-3 (1)
Hexokinase (1)
HIF (1)
IAP (1)
IGF-1R (1)
iGluR (1)
HSP (1)
Histone Demethylase (1)
ATM/ATR (1)
Beta-Secretase (1)
Bradykinin Receptor (1)
Cannabinoid Receptor (1)
CCR (1)
Caspase (1)
Antifolate (1)
ACK (1)
Akt (1)
CSF-1R (1)
CETP (1)
c-Fms (1)
CGRP Receptor (1)
DUB (1)
DNA Alkylator/Crosslinker (1)
Ephrin Receptor (1)
Epigenetic Reader Domain (1)
Ferroptosis (1)