Home Tools
Log in
Cart

FDA-Approved Drug Library

Catalog No. L4200
  Library Compound List   Excel SDF

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

In addtion, we put the compounds that should be provided in the form of dry powder together to form Part B in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L4200)

Library Composition

Antibacterial (271)
Antibiotic (265)
Autophagy (252)
Apoptosis (164)
Endogenous Metabolite (131)
Adrenergic Receptor (122)
5-HT Receptor (111)
AChR (88)
Histamine Receptor (71)
Dopamine Receptor (69)
HIV Protease (66)
COX (60)
DNA/RNA Synthesis (60)
Sodium Channel (56)
Parasite (54)
Antifungal (52)
Potassium Channel (49)
Glucocorticoid Receptor (47)
Estrogen/progestogen Receptor (39)
Calcium Channel (37)
Topoisomerase (36)
P450 (33)
Ferroptosis (32)
ribosome (29)
RAAS (27)
GABA Receptor (26)
SARS-CoV (26)
VEGFR (25)
Serotonin Transporter (25)
Mitophagy (24)
c-Kit (24)
Dehydrogenase (23)
PDE (23)
Microtubule Associated (22)
Reverse Transcriptase (22)
Nucleoside Antimetabolite/Analog (22)
Antifection (22)
HCV Protease (21)
Norepinephrine (21)
PDGFR (20)
HSV (19)
Progesterone Receptor (19)
Estrogen Receptor/ERR (18)
Reactive Oxygen Species (18)
Influenza Virus (18)
EGFR (17)
DNA Alkylator/Crosslinker (17)
PPAR (17)
Proton pump (17)
Androgen Receptor (16)
Proteasome (14)
HBV (14)
AChE (14)
Prostaglandin Receptor (14)
Carbonic Anhydrase (14)
ATPase (13)
Thrombin (13)
FLT (13)
Antifolate (12)
Opioid Receptor (12)
Virus Protease (12)
MAO (12)
MRP (11)
DHFR (11)
GNRH Receptor (11)
c-Met/HGFR (11)
Raf (11)
Adenosine Receptor (11)
ROS (11)
FGFR (11)
Phosphatase (10)
Monoamine Oxidase (10)
HDAC (10)
Src (10)
JAK (10)
iGluR (10)
c-RET (10)
NO Synthase (9)
Tyrosine Kinases (9)
NF-κB (9)
Bcr-Abl (9)
ALK (9)
Drug Metabolite (9)
Transferase (9)
TRP/TRPV Channel (9)
HMG-CoA Reductase (8)
MMP (8)
CDK (8)
Thyroid hormone receptor(THR) (8)
GluR (8)
Retinoid Receptor (8)
DNA gyrase (8)
CaMK (8)
Phospholipase (8)
PI3K (7)
Guanylate cyclase (7)
MEK (7)
P-gp (7)
ABC (7)
NMDAR (7)
DPP-4 (7)
HIF/HIF Prolyl-Hydroxylase (7)
DNA Alkylation (7)
P2Y Receptor (7)
TNF (6)
TAM Receptor (6)
Lipoxygenase (6)
mTOR (6)
CAT (6)
Factor Xa (6)
STAT (6)
PARP (6)
PKC (6)
HER (6)
SGLT (5)
S1P Receptor (5)
GPR (5)
LPL Receptor (5)
Cell wall (5)
IL Receptor (5)
TLR (5)
Neurokinin receptor (5)
Endothelin Receptor (5)
Trk receptor (5)
DNA Methyltransferase (5)
CFTR (5)
Monoamine Transporter (5)
Hedgehog/Smoothened (5)
Histone Methyltransferase (5)
Histone Demethylase (5)
Antiviral (4)
Aromatase (4)
Annexin A (4)
Reductase (4)
ROS Kinase (4)
Glutathione Peroxidase (4)
Leukotriene Receptor (4)
NADPH (4)
Ras (4)
AMPK (4)
Nrf2 (4)
ERK (4)
DNA (4)
Neprilysin (3)
BCL (3)
MT Receptor (3)
BTK (3)
NOS (3)
PAK (3)
Integrin (3)
Mitochondrial Metabolism (3)
Amino Acids and Derivatives (3)
Fatty Acid Synthase (3)
FXR (3)
Vasopressin Receptor (3)
AhR (3)
Decarboxylase (3)
Cysteine Protease (3)
CXCR (3)
Chloride channel (3)
Somatostatin (3)
CaSR (3)
Hydroxylase (3)
Smo (3)
ROCK (3)
Complement System (3)
Sigma receptor (3)
IGF-1R (3)
Beta Amyloid (2)
Thrombopoietin Receptor (2)
Beta-Secretase (2)
Aryl Hydrocarbon Receptor (2)
Serine Protease (2)
Protease-activated Receptor (2)
RSV (2)
UGT (2)
Rho (2)
Adenosine deaminase (2)
Arginase (2)
Wnt/beta-catenin (2)
Xanthine Oxidase (2)
Syk (2)
Ephrin Receptor (2)
PGE Synthase (2)
GPCR19 (2)
Integrase (2)
Interleukin (2)
IRE1 (2)
Isocitrate Dehydrogenase (IDH) (2)
Caspase (2)
LDL (2)
Lipid (2)
LTR (2)
cholecystokinin (2)
Melanocortin Receptor (2)
Melatonin Receptor (2)
CGRP Receptor (2)
HIF (2)
GST (2)
GSK-3 (2)
CRM1 (2)
Free radical scavengers (2)
CCR (2)
c-Fms (2)
Oxytocin Receptor (2)
CETP (2)
Gap Junction Protein (2)
Glutathione reductase (2)
Gamma-secretase (2)
Histone Acetyltransferase (1)
DUB (1)
FAAH (1)
ACK (1)
CSF-1R (1)
GlyT (1)
VDA (1)
TGF-beta/Smad (1)
GluCls (1)
Akt (1)
Tyrosinase (1)
Glucosidase (1)
HSP (1)
GRK (1)
Telomerase (1)
Angiotensin-converting Enzyme (ACE) (1)
CRISPR/Cas9 (1)
Epigenetic Reader Domain (1)
P2X Receptor (1)
Phosphorylase (1)
OX Receptor (1)
PKM (1)
Platelet aggregation (1)
PLK (1)
OAT (1)
Bradykinin Receptor (1)
NPC1L1 (1)
NOD-like Receptor (NLR) (1)
Pyroptosis (1)
Hydrogenase (1)
ATP Citrate Lyase (1)
Na-K-Cl cotransporter (1)
RAR/RXR  (1)
NADPH-oxidase (1)
MTH1 (1)
Chk (1)
MAPK (1)
ROR (1)
IκB/IKK (1)
Sirtuin (1)
IAP (1)
YAP (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE