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Compound Libraries Drug Repurposing Library

Drug Repurposing Library

Catalog No. L9200
  Library Compound List   Excel SDF

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

The Drug Repurposing Library by TargetMol, containing 3512 approved and clinical drugs, which have undergone extensive preclinical studies and have well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization, is a good tool for drug repurposing and cell induction.

In addtion, we provide the peptides and other drug molecules with low solution stability in the form of dry powder (set as Part B) in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 28119.00
250 μL * 10 mM (in DMSO) 49534.00
1 mg 49534.00
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Product Description

  • A unique collection of 3512 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • All approved drugs collected in this library are approved by Food and Drug Administration (FDA), the European Medicine Agency (EMA), or China Food and Drug Administration (CFDA), or included in the US Pharmacopeia (USP) Dictionary, the British Pharmacopoeia (BP), the European Pharmacopoeia (EP), the Japanese Pharmacopoeia (JP), or Chinese Pharmacopoeia (CP) Dictionary;
  • Covers various research areas, such as cancer, cardiovascular disease, immunology, respiratory system, etc.
  • Covers various targets, such as 5-HT Receptor, Sodium Channel, p38 MAPK, PI3K, MEK, etc.
  • Detailed compound information with structure, target, activity, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L9200)

Library Composition

Adrenergic Receptor (144)
5-HT Receptor (143)
AChR (134)
Antibiotic (114)
COX (104)
Antibacterial (101)
Dopamine Receptor (100)
DNA/RNA Synthesis (71)
Histamine Receptor (70)
Sodium Channel (70)
VEGFR (59)
Calcium Channel (55)
Estrogen/progestogen Receptor (54)
Potassium Channel (54)
PI3K (51)
Endogenous Metabolite (51)
Topoisomerase (49)
PDE (48)
Glucocorticoid Receptor (47)
Autophagy (47)
EGFR (45)
GABA Receptor (44)
Dehydrogenase (43)
HIV Protease (40)
JAK (39)
PDGFR (38)
HDAC (38)
FGFR (36)
CDK (36)
RAAS (36)
PPAR (35)
c-Kit (35)
FLT (35)
GR (34)
Microtubule Associated (33)
Vitamin (33)
P450 (32)
Bcr-Abl (31)
Androgen Receptor (29)
Src (29)
mTOR (29)
NF-κB (28)
Antifungal (28)
c-Met/HGFR (28)
HCV Protease (25)
MAO (25)
ribosome (25)
Tyrosine Kinases (24)
Raf (22)
Opioid Receptor (22)
NMDAR (22)
Norepinephrine (22)
Carbonic Anhydrase (22)
Antifection (21)
Prostaglandin Receptor (21)
TNF (20)
ATPase (19)
DNA Alkylation (19)
Akt (18)
Antioxidant (17)
ROS (17)
MEK (17)
HSP (16)
Reverse Transcriptase (16)
Adenosine Receptor (16)
BTK (16)
GPR (16)
GluR (16)
Epigenetic Reader Domain (15)
ALK (15)
Antiviral (15)
PKC (15)
PARP (15)
IL Receptor (15)
p38 MAPK (14)
Parasite (14)
DPP-4 (14)
Thyroid hormone receptor(THR) (14)
TAM Receptor (13)
DNA-PK (13)
c-RET (13)
HER (13)
Retinoid Receptor (13)
MRP (13)
Proton pump (12)
GSK-3 (12)
Amino Acids and Derivatives (12)
Aurora Kinase (12)
Thrombin (12)
Transferase (12)
TRP/TRPV Channel (11)
Apoptosis (11)
HIF (11)
DNA gyrase (11)
STAT (11)
NADPH (11)
MMP (11)
Influenza Virus (10)
Lipoxygenase (10)
S1P Receptor (10)
Proteasome (10)
CXCR (10)
HBV (10)
Glucokinase (10)
Chk (10)
Trk receptor (10)
Syk (10)
CFTR (9)
Beta Amyloid (9)
CaMK (9)
AMPK (9)
Gamma-secretase (9)
Hedgehog/Smoothened (9)
Endothelin Receptor (9)
PKA (9)
PLK (9)
Phospholipase (9)
Serine Protease (9)
SGLT (9)
Integrin (9)
HMG-CoA Reductase (8)
S6 Kinase (8)
ROCK (8)
ERK (8)
FAK (8)
CCR (8)
CSF-1R (8)
FXR (8)
BCL (8)
Cannabinoid Receptor (8)
Caspase (7)
ABC (7)
Aromatase (7)
ATM/ATR (7)
DHFR (7)
Sigma receptor (7)
P-gp (7)
Phosphatase (7)
p53 (7)
P2 Receptor (7)
HSV (7)
Hydroxylase (7)
IDO (7)
JNK (7)
TLR (7)
Tyrosinase (7)
Wnt/beta-catenin (7)
Vasopressin Receptor (6)
TGF-beta/Smad (6)
IκB/IKK (6)
LTR (6)
IGF-1R (6)
IAP (6)
Histone Demethylase (6)
Histone Methyltransferase (6)
NOS (6)
Nucleoside Antimetabolite/Analog (6)
Reductase (6)
Cysteine Protease (6)
Factor Xa (6)
AhR (6)
CAT (6)
Chloride channel (6)
CETP (5)
c-Fms (5)
Casein Kinase (5)
BACE (5)
DNA Methyltransferase (5)
GNRH Receptor (5)
Ras (5)
Sirtuin (5)
Serotonin Transporter (5)
Pim (5)
MPO (5)
OX Receptor (5)
Neurokinin receptor (5)
Mdm2 (5)
Mitochondrial Metabolism (5)
UGT (5)
Liver X Receptor (4)
Kinesin (4)
Monoamine Transporter (4)
NOD (4)
GHSR (4)
Guanylate cyclase (4)
HIF/HIF Prolyl-Hydroxylase (4)
Fatty Acid Synthase (4)
FAAH (4)
DprE1 (4)
Aminopeptidase (4)
Annexin A (4)
ATP Citrate Lyase (3)
Acyltransferase (3)
CaSR (3)
Cell wall (3)
cholecystokinin (3)
Ferroptosis (3)
Decarboxylase (3)
GST (3)
Gap Junction Protein (3)
Free radical scavengers (3)
GPCR19 (3)
GlyT (3)
Neuropeptide Y Receptor (3)
Nrf2 (3)
Monocarboxylate transporter (3)
NADPH-oxidase (3)
Na-K-Cl cotransporter (3)
Lipid (3)
PAK (3)
PDK (3)
ROR (3)
Rho (3)
Telomerase (3)
Tie-2 (2)
VDA (2)
RSV (2)
PYK2 (2)
SARS-CoV (2)
Serine/threonin kinase (2)
OAT (2)
PKM (2)
Protease-activated Receptor (2)
LPA Receptor (2)
KSP (2)
LDL (2)
Lipase (2)
MAPK (2)
IRAK (2)
NAMPT (2)
Neprilysin (2)
MT Receptor (2)
Monoamine Oxidase (2)
Melatonin Receptor (2)
Glutathione Peroxidase (2)
Glutathione reductase (2)
Glucagon Receptor (2)
GluCls (2)
Hexokinase (2)
CRFR (2)
CRM1 (2)
DNA (2)
DUB (2)
E1/E2/E3 Enzyme (2)
Ephrin Receptor (2)
c-Myc (2)
Complement System (2)
ACAT (2)
Acetyl-CoA Carboxylase (2)
AChE (2)
advanced glycation end products (2)
Antifolate (2)
Anti-infection (1)
Anion Exchanger (1)
ASK (1)
Apoptosis inducer (1)
Arginase (1)
ACK (1)
CPT (1)
CGRP Receptor (1)
cAMP (1)
Beta-Secretase (1)
Bradykinin Receptor (1)
Electron transport (1)
Estrogen Receptor/ERR (1)
Dehydrogenase inhibitor (1)
Discoidin Domain Receptor (DDR) (1)
DNA Alkylator/Crosslinker (1)
Hck (1)
GSNOR (1)
GRK (1)
FLAP (1)
MELK (1)
MNK (1)
Myosin (1)
N-Acetylglucosaminyltransferase (1)
NPC1L1 (1)
OXPHOS (1)
Oxytocin Receptor (1)
NKCC (1)
NOD-like Receptor (NLR) (1)
NO Synthase (1)
Isocitrate Dehydrogenase (IDH) (1)
Integrase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Hydrogenase (1)
lysosomal autophagy (1)
Mitophagy (1)
MLK (1)
Porcupine (1)
Progesterone Receptor (1)
Platelet aggregation (1)
P2X Receptor (1)
p97 (1)
PAFR (1)
PAI-1 (1)
PED (1)
PGE Synthase (1)
Smo (1)
SGK (1)
Somatostatin (1)
Stemness kinase (1)
STING (1)
Survivin (1)
RAR/RXR (1)
Reactive Oxygen Species (1)
RIP kinase (1)
Xanthine Oxidase (1)
Wee1 (1)
Thrombopoietin Receptor (1)
Thioredoxin (1)
transporter (1)