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Compound Libraries Clinical Compound Library

Clinical Compound Library

Catalog No. L3400
  Library Compound List   Excel SDF

Clinical compound library is a collection of 1487 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 17640.00
250 μL * 10 mM (in DMSO) 29010.00
1 mg 29010.00
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Product Description

  • A unique collection of 1487 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging and Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice.
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Library Composition

PI3K (41)
VEGFR (36)
CDK (35)
EGFR (34)
JAK (28)
FLT (26)
FGFR (22)
mTOR (22)
c-Met/HGFR (20)
PDGFR (20)
Bcr-Abl (18)
c-Kit (17)
HDAC (17)
Src (17)
Aurora Kinase (16)
5-HT Receptor (16)
Akt (15)
p38 MAPK (15)
Tyrosine Kinases (14)
DNA/RNA Synthesis (14)
HSP (14)
GSK-3 (13)
ALK (12)
DNA-PK (11)
Epigenetic Reader Domain (11)
HER (11)
Microtubule Associated (11)
PKC (11)
Raf (11)
PARP (10)
GPR (10)
COX (10)
AChR (10)
Androgen Receptor (10)
Chk (9)
Estrogen/progestogen Receptor (9)
Histamine Receptor (9)
MEK (9)
PPAR (9)
Syk (9)
TAM Receptor (9)
Dehydrogenase (8)
BTK (8)
c-RET (7)
ERK (7)
Histone Methyltransferase (7)
HIF (7)
IDO (7)
HCV Protease (7)
GluR (7)
Trk receptor (7)
PDE (7)
P450 (6)
PDK (6)
Phospholipase (6)
Pim (6)
PKA (6)
Potassium Channel (6)
TLR (6)
Gamma-secretase (6)
IGF-1R (6)
Mdm2 (6)
NF-κB (6)
FAK (6)
Dopamine Receptor (6)
Beta Amyloid (6)
ATPase (6)
Adenosine Receptor (6)
Adrenergic Receptor (5)
Antibacterial (5)
Calcium Channel (5)
Cannabinoid Receptor (5)
Casein Kinase (5)
Caspase (5)
CCR (5)
FAAH (5)
CSF-1R (5)
CXCR (5)
Cysteine Protease (5)
c-Fms (5)
BCL (5)
MMP (5)
IκB/IKK (5)
IL Receptor (5)
HIV Protease (5)
GABA Receptor (5)
Transferase (5)
TRP/TRPV Channel (5)
STAT (5)
ROS (5)
RAAS (5)
Prostaglandin Receptor (5)
p53 (5)
P2 Receptor (4)
PLK (4)
Proteasome (4)
ROCK (4)
Sigma receptor (4)
Sirtuin (4)
Sodium Channel (4)
S1P Receptor (4)
S6 Kinase (4)
Serine Protease (4)
TGF-beta/Smad (4)
IAP (4)
LPA Receptor (4)
Antiviral (4)
ATM/ATR (4)
BACE (3)
Carbonic Anhydrase (3)
Antibiotic (3)
AMPK (3)
CETP (3)
CFTR (3)
cholecystokinin (3)
DNA Alkylation (3)
CRM1 (3)
DUB (3)
Liver X Receptor (3)
Kinesin (3)
NADPH (3)
NMDAR (3)
OX Receptor (3)
HSV (3)
Hydroxylase (3)
Histone Demethylase (3)
HIF/HIF Prolyl-Hydroxylase (3)
Hedgehog/Smoothened (3)
Glucokinase (3)
Tie-2 (3)
Wnt/beta-catenin (3)
transporter (3)
TNF (3)
Opioid Receptor (3)
PAK (2)
P-gp (2)
Phosphatase (2)
PYK2 (2)
Ras (2)
Retinoid Receptor (2)
Reverse Transcriptase (2)
UGT (2)
Vasopressin Receptor (2)
Topoisomerase (2)
Vitamin (2)
SGLT (2)
FXR (2)
Glucocorticoid Receptor (2)
Integrin (2)
Norepinephrine (2)
NOS (2)
NAMPT (2)
KSP (2)
Lipoxygenase (2)
JNK (2)
LTR (2)
DprE1 (2)
Endothelin Receptor (2)
Antioxidant (2)
Autophagy (2)
ATP Citrate Lyase (1)
Apoptosis inducer (1)
ASK (1)
CaMK (1)
Bombesin Receptor (1)
ACAT (1)
Antifection (1)
Antifungal (1)
advanced glycation end products (1)
AhR (1)
Amino Acids and Derivatives (1)
Aminopeptidase (1)
Ephrin Receptor (1)
Ferroptosis (1)
DYRK (1)
DPP-4 (1)
DNA Methyltransferase (1)
CGRP Receptor (1)
cell cycle arrest (1)
lysosomal autophagy (1)
MAO (1)
MELK (1)
LDL (1)
LHRH (1)
Neurokinin 1 (1)
NADPH-oxidase (1)
MNK (1)
Monocarboxylate transporter (1)
MLK (1)
Nrf2 (1)
OAT (1)
NOD (1)
Influenza Virus (1)
GlyT (1)
GNRH Receptor (1)
GR (1)
GSNOR (1)
HBV (1)
Hck (1)
Survivin (1)
Thioredoxin (1)
Thrombin (1)
Thyroid hormone receptor(THR) (1)
SGK (1)
Wee1 (1)
VDA (1)
TOPK (1)
Rho (1)
Reductase (1)
Proton pump (1)
Porcupine (1)
Protease-activated Receptor (1)
Platelet aggregation (1)
PED (1)
PERK (1)
p97 (1)
PAFR (1)
PAI-1 (1)