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Compound Libraries Clinical Compound Library

Clinical Compound Library

Catalog No. L3400
  Library Compound List   Excel SDF

Clinical compound library is a collection of 2500 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 29724.00
250 μL * 10 mM (in DMSO) 48780.00
1 mg 48780.00
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Product Description

  • A unique collection of 2500 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L3400)

Library Composition

5-HT Receptor (101)
Adrenergic Receptor (83)
AChR (81)
Dopamine Receptor (70)
COX (60)
DNA/RNA Synthesis (58)
VEGFR (53)
Antibacterial (52)
Antibiotic (52)
PI3K (49)
Sodium Channel (46)
Histamine Receptor (42)
Potassium Channel (41)
Calcium Channel (38)
Estrogen/progestogen Receptor (37)
PDE (37)
JAK (36)
Endogenous Metabolite (36)
EGFR (35)
Glucocorticoid Receptor (35)
HDAC (34)
Dehydrogenase (34)
Topoisomerase (34)
CDK (33)
HIV Protease (33)
PDGFR (33)
FLT (32)
FGFR (31)
GABA Receptor (29)
RAAS (29)
mTOR (29)
c-Kit (28)
Src (27)
PPAR (26)
Microtubule Associated (26)
c-Met/HGFR (26)
Autophagy (26)
Androgen Receptor (24)
P450 (24)
Bcr-Abl (23)
GR (23)
HCV Protease (22)
Tyrosine Kinases (22)
NF-κB (19)
Raf (19)
DNA Alkylation (18)
Vitamin (18)
Carbonic Anhydrase (17)
Akt (17)
Norepinephrine (17)
MEK (17)
NMDAR (16)
ROS (16)
Prostaglandin Receptor (16)
Antifection (16)
BTK (16)
ALK (15)
Epigenetic Reader Domain (15)
GPR (15)
HSP (15)
Opioid Receptor (14)
Adenosine Receptor (14)
Antifungal (14)
Antioxidant (14)
ATPase (14)
TNF (14)
GluR (13)
DNA-PK (13)
ribosome (13)
Reverse Transcriptase (13)
IL Receptor (13)
Retinoid Receptor (12)
TAM Receptor (12)
PARP (12)
Aurora Kinase (12)
Antiviral (11)
Apoptosis (11)
DPP-4 (11)
c-RET (11)
HER (11)
p38 MAPK (11)
Transferase (11)
Trk receptor (10)
STAT (10)
MAO (10)
MRP (10)
HIF (10)
GSK-3 (10)
HBV (10)
Glucokinase (10)
Gamma-secretase (10)
CXCR (9)
S1P Receptor (9)
Proteasome (9)
PLK (9)
TRP/TRPV Channel (9)
Syk (9)
Thyroid hormone receptor(THR) (9)
Thrombin (8)
PKC (8)
SGLT (8)
NADPH (8)
Integrin (8)
CSF-1R (8)
ERK (8)
Endothelin Receptor (8)
Hedgehog/Smoothened (8)
Beta Amyloid (8)
CFTR (8)
Chk (8)
CCR (7)
BCL (7)
Influenza Virus (7)
IDO (7)
Hydroxylase (7)
HMG-CoA Reductase (7)
MMP (7)
S6 Kinase (7)
P-gp (7)
Proton pump (7)
Wnt/beta-catenin (7)
TLR (6)
Phosphatase (6)
Parasite (6)
P2 Receptor (6)
p53 (6)
Sigma receptor (6)
Serine Protease (6)
Nucleoside Antimetabolite/Analog (6)
HSV (6)
IGF-1R (6)
Lipoxygenase (6)
JNK (6)
Cannabinoid Receptor (6)
Caspase (6)
ATM/ATR (6)
Amino Acids and Derivatives (6)
AhR (6)
AMPK (6)
FXR (6)
FAK (6)
DHFR (6)
DNA gyrase (5)
DNA Methyltransferase (5)
GNRH Receptor (5)
CAT (5)
CETP (5)
Casein Kinase (5)
LTR (5)
IκB/IKK (5)
Mdm2 (5)
IAP (5)
Histone Methyltransferase (5)
NOS (5)
Neurokinin receptor (5)
Mitochondrial Metabolism (5)
Sirtuin (5)
ROCK (5)
Ras (5)
Phospholipase (5)
Pim (5)
PKA (5)
Vasopressin Receptor (5)
OX Receptor (4)
Reductase (4)
TGF-beta/Smad (4)
MPO (4)
Liver X Receptor (4)
Kinesin (4)
CaMK (4)
BACE (4)
c-Fms (4)
Acyltransferase (4)
HIF/HIF Prolyl-Hydroxylase (4)
Histone Demethylase (4)
Guanylate cyclase (4)
Cysteine Protease (4)
Fatty Acid Synthase (4)
FAAH (4)
Factor Xa (4)
Ferroptosis (3)
DprE1 (3)
Decarboxylase (3)
Gap Junction Protein (3)
GHSR (3)
Free radical scavengers (3)
ABC (3)
ATP Citrate Lyase (3)
Arginase (3)
Aromatase (3)
Chloride channel (3)
Nrf2 (3)
Neuropeptide Y Receptor (3)
NADPH-oxidase (3)
Na-K-Cl cotransporter (3)
MT Receptor (3)
Serotonin Transporter (3)
Rho (3)
ROR (3)
Tyrosinase (3)
UGT (3)
VDA (2)
Tie-2 (2)
SARS-CoV (2)
RSV (2)
Telomerase (2)
PAK (2)
PDK (2)
PYK2 (2)
Melatonin Receptor (2)
NAMPT (2)
Neprilysin (2)
OAT (2)
KSP (2)
LDL (2)
LPA Receptor (2)
MAPK (2)
cholecystokinin (2)
c-Myc (2)
Complement System (2)
CaSR (2)
Annexin A (2)
Antifolate (2)
ACAT (2)
Acetyl-CoA Carboxylase (2)
Aminopeptidase (2)
Glucagon Receptor (2)
GPCR19 (2)
Glutathione Peroxidase (2)
GlyT (2)
GST (2)
CRFR (2)
CRM1 (2)
DNA (2)
DUB (2)
E1/E2/E3 Enzyme (2)
Ephrin Receptor (2)
Electron transport (1)
Discoidin Domain Receptor (DDR) (1)
DNA Alkylator/Crosslinker (1)
CPT (1)
Dehydrogenase inhibitor (1)
Hck (1)
GSNOR (1)
GRK (1)
Hexokinase (1)
GluCls (1)
FLAP (1)
advanced glycation end products (1)
ACK (1)
Anti-infection (1)
Anion Exchanger (1)
ASK (1)
Apoptosis inducer (1)
Beta-Secretase (1)
Bradykinin Receptor (1)
Cell wall (1)
CGRP Receptor (1)
lysosomal autophagy (1)
LHRH (1)
Lipase (1)
Lipid (1)
Hydrogenase (1)
iGluR (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Integrase (1)
IRAK (1)
Isocitrate Dehydrogenase (IDH) (1)
NPC1L1 (1)
NKCC (1)
Myosin (1)
N-Acetylglucosaminyltransferase (1)
NO Synthase (1)
NOD (1)
NOD-like Receptor (NLR) (1)
MELK (1)
Mitophagy (1)
MLK (1)
MNK (1)
Monoamine Oxidase (1)
Monoamine Transporter (1)
Monocarboxylate transporter (1)
Protease-activated Receptor (1)
Porcupine (1)
Progesterone Receptor (1)
PKM (1)
PGE Synthase (1)
OXPHOS (1)
Oxytocin Receptor (1)
p97 (1)
PAFR (1)
PAI-1 (1)
Thioredoxin (1)
Stemness kinase (1)
STING (1)
Survivin (1)
SGK (1)
Somatostatin (1)
Smo (1)
RIP kinase (1)
Reactive Oxygen Species (1)
RAR/RXR (1)
transporter (1)
Wee1 (1)
Xanthine Oxidase (1)