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Compound Libraries Bioactive Lipid Compound Library

Bioactive Lipid Compound Library

Catalog No. L7000
  Library Compound List   Excel SDF

Bioactive lipids have been shown to provide health benefits either through modification of tissue fatty acid composition or induction of cell signaling pathways, due to their pivotal role in immune regulation, inflammation, and maintenance of tissue homeostasis. While some health benefits are derived from consumption of short to medium-chain fatty acids, evidence suggests that the polyunsaturated fatty acids (PUFAs) are the most important bioactive lipids. PUFAs are found mostly in plant seed oils and are important substrates for the biosynthesis of cellular hormones (eicosanoids) and other signaling compounds that modulate human health. The beneficial health effects of PUFAs seem to be dependent on their isomer configuration as the cis-isomer is the predominant bioactive form which enhances membrane fluidity when incorporated into cells. Increased membrane fluidity enhances cell to cell communication and helps maintain normal homeostasis or prevent the development of metabolic disorders.

The TargetMol’s Bioactive Lipid Inhibitor Library, a unique collection of 280 bioactive lipids related compounds, can be used for research in bioactive lipids, and high throughput screening (HTS) and high content screening (HCS).

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 4675.00
250 μL * 10 mM (in DMSO) 7800.00
1 mg 7800.00
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Product Description

  • A unique collection of 280 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, HETEs deHETEs, hepoxilins, Polyunsaturated fatty acids, Leukotrienes, lipoxins, LPA & phosphatidic acids, Octadecanoids, PAFs, Prostaglandins & thromboxanes, Retinoids, vitamin D metabolites, Sphingolipids, etc.;
  • Targets include GPCR, HDAC, PPAR, DNA Alkylating, EGFR, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging and Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice.
Request Library Compound List (L7000)

Library Composition

PDE (40)
Phospholipase (16)
MAO (14)
COX (14)
HMG-CoA Reductase (9)
Lipase (8)
PPAR (8)
Thrombin (8)
Vitamin (7)
Retinoid Receptor (7)
Lipid (7)
Lipoxygenase (7)
FXR (7)
Factor Xa (6)
Cannabinoid Receptor (6)
AhR (6)
P450 (6)
AChR (5)
Fatty Acid Synthase (5)
CETP (4)
Prostaglandin Receptor (4)
NF-κB (4)
Liver X Receptor (3)
PLK (3)
ACAT (3)
Adrenergic Receptor (3)
DNA/RNA Synthesis (3)
HDAC (3)
TNF (3)
LDL (2)
Sodium Channel (2)
Histamine Receptor (2)
GPR (2)
Glucocorticoid Receptor (2)
Dehydrogenase (2)
Adenosine Receptor (2)
Bcr-Abl (2)
Calcium Channel (2)
Potassium Channel (2)
PED (2)
MPO (2)
mTOR (1)
NADPH (1)
NADPH-oxidase (1)
NMDAR (1)
Opioid Receptor (1)
MMP (1)
Monocarboxylate transporter (1)
LPA Receptor (1)
LTR (1)
lysosomal autophagy (1)
Hydroxylase (1)
IAP (1)
IL Receptor (1)
IκB/IKK (1)
Phosphatase (1)
Serine Protease (1)
Sirtuin (1)
PAI-1 (1)
PDGFR (1)
Phosphorylase (1)
PI3K (1)
PKA (1)
PKM (1)
Platelet aggregation (1)
Casein Kinase (1)
Chloride channel (1)
c-Met/HGFR (1)
c-RET (1)
Cysteine Protease (1)
5-HT Receptor (1)
ABC (1)
AMPK (1)
Autophagy (1)
DNA (1)
DNA Alkylation (1)
Dopamine Receptor (1)
Estrogen/progestogen Receptor (1)
FAAH (1)
GluR (1)
GPCR19 (1)
GABA Receptor (1)
GR (1)
Histone Demethylase (1)
TGF-beta/Smad (1)
Topoisomerase (1)
Transferase (1)
Tyrosinase (1)
UGT (1)
VEGFR (1)
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