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Compound Libraries Anti-cancer Clinical Compound Library

Anti-cancer Clinical Compound Library

Catalog No. L2120
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 594 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 9890.00
250 μL * 10 mM (in DMSO) 16310.00
1 mg 16310.00
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Product Description

  • A unique collection of 594 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging and Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice.
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Library Composition

PI3K (38)
VEGFR (35)
CDK (34)
EGFR (33)
FLT (25)
FGFR (23)
JAK (21)
mTOR (20)
PDGFR (20)
c-Met/HGFR (20)
Bcr-Abl (18)
Aurora Kinase (16)
c-Kit (16)
Src (16)
HSP (14)
HDAC (13)
Akt (13)
ALK (12)
HER (11)
DNA/RNA Synthesis (11)
Raf (11)
Tyrosine Kinases (11)
Microtubule Associated (10)
DNA-PK (10)
Epigenetic Reader Domain (10)
Chk (10)
TAM Receptor (9)
GSK-3 (8)
MEK (8)
IGF-1R (8)
PKC (8)
PDK (7)
PARP (7)
p38 MAPK (7)
Histone Methyltransferase (7)
Trk receptor (7)
ERK (6)
Estrogen/progestogen Receptor (6)
c-RET (6)
BTK (6)
IDO (6)
Mdm2 (6)
Pim (6)
PKA (5)
STAT (5)
Syk (5)
MMP (5)
NF-κB (5)
BCL (5)
Casein Kinase (5)
c-Fms (5)
Androgen Receptor (5)
FAK (5)
CSF-1R (5)
CXCR (4)
IAP (4)
ATM/ATR (4)
COX (4)
P450 (4)
p53 (4)
ROS (4)
S6 Kinase (4)
PLK (4)
Proteasome (4)
LPA Receptor (3)
IκB/IKK (3)
Kinesin (3)
Caspase (3)
Carbonic Anhydrase (3)
Adenosine Receptor (3)
Histone Demethylase (3)
HIF (3)
Gamma-secretase (3)
Hedgehog/Smoothened (3)
Dehydrogenase (3)
DNA Alkylation (3)
DUB (3)
transporter (3)
Wnt/beta-catenin (3)
Topoisomerase (3)
Tie-2 (3)
TLR (3)
TNF (2)
Transferase (2)
TGF-beta/Smad (2)
UGT (2)
Cysteine Protease (2)
Ephrin Receptor (2)
HCV Protease (2)
Histamine Receptor (2)
ATPase (2)
Beta Amyloid (2)
CRM1 (2)
CFTR (2)
cholecystokinin (2)
KSP (2)
IL Receptor (2)
Integrin (2)
Lipoxygenase (2)
NAMPT (2)
PAK (2)
PYK2 (2)
PPAR (2)
Prostaglandin Receptor (2)
P-gp (2)
Phospholipase (2)
PDE (2)
Ras (2)
Retinoid Receptor (2)
Sirtuin (2)
ROCK (2)
Survivin (1)
Sodium Channel (1)
S1P Receptor (1)
Reverse Transcriptase (1)
Rho (1)
Serine Protease (1)
SGK (1)
Sigma receptor (1)
PERK (1)
Porcupine (1)
Potassium Channel (1)
P2 Receptor (1)
p97 (1)
PAFR (1)
NOS (1)
Nrf2 (1)
Opioid Receptor (1)
MNK (1)
Monocarboxylate transporter (1)
NADPH (1)
lysosomal autophagy (1)
MELK (1)
MLK (1)
LDL (1)
JNK (1)
Calcium Channel (1)
CaMK (1)
CCR (1)
cell cycle arrest (1)
Autophagy (1)
AChR (1)
Antifection (1)
Apoptosis inducer (1)
ASK (1)
Aminopeptidase (1)
AMPK (1)
HIV Protease (1)
HSV (1)
Glucokinase (1)
GNRH Receptor (1)
Hck (1)
GABA Receptor (1)
Ferroptosis (1)
DNA Methyltransferase (1)
DPP-4 (1)
VDA (1)
Wee1 (1)
Thioredoxin (1)
TOPK (1)
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