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Compound Libraries Anti-cancer Clinical Compound Library

Anti-cancer Clinical Compound Library

Catalog No. L2120
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1776 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 21115.00
250 μL * 10 mM (in DMSO) 34652.00
1 mg 34652.00
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Product Description

  • A unique collection of 1776 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2120)

Library Composition

DNA/RNA Synthesis (59)
COX (58)
AChR (55)
VEGFR (55)
PI3K (48)
EGFR (38)
CDK (35)
JAK (35)
PDGFR (34)
Dehydrogenase (34)
HDAC (34)
FLT (33)
Estrogen/progestogen Receptor (33)
Topoisomerase (33)
Potassium Channel (33)
FGFR (31)
c-Kit (31)
Adrenergic Receptor (30)
Glucocorticoid Receptor (29)
mTOR (29)
c-Met/HGFR (28)
Microtubule Associated (27)
PPAR (27)
Src (27)
Bcr-Abl (26)
PDE (25)
Sodium Channel (24)
RAAS (23)
Autophagy (22)
GR (22)
Antibacterial (21)
Androgen Receptor (21)
Tyrosine Kinases (21)
P450 (20)
GABA Receptor (20)
DNA Alkylation (18)
Raf (18)
NF-κB (17)
Akt (17)
Antibiotic (16)
Antifection (16)
Carbonic Anhydrase (16)
MEK (16)
ALK (15)
Endogenous Metabolite (15)
Epigenetic Reader Domain (15)
HSP (14)
IL Receptor (14)
BTK (14)
TAM Receptor (14)
PARP (13)
c-RET (13)
Calcium Channel (12)
ATPase (12)
Aurora Kinase (12)
HIF (12)
HER (12)
HIV Protease (12)
DNA-PK (12)
TNF (12)
Retinoid Receptor (12)
Reverse Transcriptase (12)
p38 MAPK (11)
MRP (11)
GPR (11)
GSK-3 (10)
Apoptosis (10)
Adenosine Receptor (10)
CXCR (10)
Integrin (10)
MAO (10)
STAT (10)
Trk receptor (10)
Vitamin (9)
Syk (9)
Thrombin (9)
ROS (9)
PKC (9)
PLK (9)
Gamma-secretase (9)
ERK (8)
Hedgehog/Smoothened (8)
CSF-1R (8)
Chk (8)
Proteasome (8)
S6 Kinase (8)
Transferase (8)
TRP/TRPV Channel (7)
Wnt/beta-catenin (7)
NADPH (7)
P-gp (7)
BCL (7)
CCR (7)
Amino Acids and Derivatives (7)
IDO (7)
DHFR (7)
FAK (6)
HSV (6)
HMG-CoA Reductase (6)
HCV Protease (6)
AMPK (6)
ATM/ATR (6)
Caspase (6)
Antiviral (6)
Beta Amyloid (6)
CFTR (6)
NOS (6)
JNK (6)
S1P Receptor (6)
Prostaglandin Receptor (6)
PKA (5)
Serine Protease (5)
Sirtuin (5)
TLR (5)
Lipoxygenase (5)
IκB/IKK (5)
Mdm2 (5)
NMDAR (5)
Nucleoside Antimetabolite/Analog (5)
Phospholipase (5)
Parasite (5)
p53 (5)
Casein Kinase (5)
Antifungal (5)
AhR (5)
HBV (5)
Hydroxylase (5)
IGF-1R (5)
Glucokinase (5)
DNA gyrase (5)
DNA Methyltransferase (5)
GluR (4)
Fatty Acid Synthase (4)
IAP (4)
HIF/HIF Prolyl-Hydroxylase (4)
Histamine Receptor (4)
Histone Demethylase (4)
Antioxidant (4)
CAT (4)
Cysteine Protease (4)
c-Fms (4)
Pim (4)
MPO (4)
Opioid Receptor (4)
Liver X Receptor (4)
TGF-beta/Smad (4)
ROCK (4)
ribosome (4)
Proton pump (4)
Reductase (3)
Ras (3)
ROR (3)
SGLT (3)
Telomerase (3)
UGT (3)
LTR (3)
LDL (3)
Nrf2 (3)
Na-K-Cl cotransporter (3)
Phosphatase (3)
PAK (3)
CETP (3)
CaMK (3)
ATP Citrate Lyase (3)
Arginase (3)
Aromatase (3)
BACE (3)
ABC (3)
Annexin A (3)
Aminopeptidase (3)
Histone Methyltransferase (3)
GNRH Receptor (3)
Free radical scavengers (3)
Factor Xa (3)
DprE1 (3)
DUB (2)
E1/E2/E3 Enzyme (2)
Dopamine Receptor (2)
DPP-4 (2)
Ferroptosis (2)
DNA (2)
Ephrin Receptor (2)
Gap Junction Protein (2)
GlyT (2)
GPCR19 (2)
ACAT (2)
Acyltransferase (2)
Antifolate (2)
Cannabinoid Receptor (2)
CaSR (2)
cholecystokinin (2)
c-Myc (2)
Decarboxylase (2)
CRM1 (2)
NAMPT (2)
P2 Receptor (2)
MAPK (2)
Kinesin (2)
KSP (2)
Influenza Virus (2)
Mitochondrial Metabolism (2)
Vasopressin Receptor (2)
VDA (2)
Tyrosinase (2)
Thyroid hormone receptor(THR) (2)
Tie-2 (2)
Rho (2)
PYK2 (2)
Protease-activated Receptor (2)
Porcupine (1)
PKM (1)
RAR/RXR (1)
Reactive Oxygen Species (1)
RIP kinase (1)
Smo (1)
Somatostatin (1)
Serotonin Transporter (1)
SGK (1)
Thioredoxin (1)
transporter (1)
Stemness kinase (1)
STING (1)
Survivin (1)
Wee1 (1)
Xanthine Oxidase (1)
Mitophagy (1)
MLK (1)
MMP (1)
MNK (1)
Monoamine Transporter (1)
Monocarboxylate transporter (1)
Melatonin Receptor (1)
MELK (1)
NADPH-oxidase (1)
MT Receptor (1)
MTH1 (1)
Integrase (1)
Isocitrate Dehydrogenase (IDH) (1)
LHRH (1)
Lipid (1)
lysosomal autophagy (1)
OXPHOS (1)
OAT (1)
Neurokinin receptor (1)
NKCC (1)
NOD-like Receptor (NLR) (1)
Norepinephrine (1)
NPC1L1 (1)
p97 (1)
PAI-1 (1)
PDK (1)
Dehydrogenase inhibitor (1)
CPT (1)
Cell wall (1)
Beta-Secretase (1)
Apoptosis inducer (1)
ASK (1)
5-HT Receptor (1)
ACK (1)
Hck (1)
FXR (1)
GST (1)
Guanylate cyclase (1)
Hexokinase (1)
Hydrogenase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
GHSR (1)
Glutathione Peroxidase (1)
Discoidin Domain Receptor (DDR) (1)
DNA Alkylator/Crosslinker (1)
Endothelin Receptor (1)
Electron transport (1)