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Compound Libraries Anti-cancer Approved drug Library

Anti-cancer Approved drug Library

Catalog No. L2110
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1400 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 9731.00
250 μL * 10 mM (in DMSO) 15960.00
1 mg 15960.00
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Product Description

  • A unique collection of 1400 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or CFDA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2110)

Library Composition

AChR (86)
COX (85)
Adrenergic Receptor (58)
DNA/RNA Synthesis (57)
Estrogen/progestogen Receptor (46)
Histamine Receptor (42)
Potassium Channel (40)
Antibacterial (39)
Topoisomerase (38)
Autophagy (32)
Glucocorticoid Receptor (32)
PDE (30)
Sodium Channel (28)
Antibiotic (28)
Dehydrogenase (27)
RAAS (26)
PPAR (25)
GR (25)
GABA Receptor (24)
VEGFR (24)
Microtubule Associated (23)
EGFR (22)
c-Kit (20)
Antifection (20)
PDGFR (19)
P450 (19)
Carbonic Anhydrase (18)
Vitamin (17)
NF-κB (16)
Androgen Receptor (16)
Bcr-Abl (15)
Calcium Channel (15)
MAO (15)
HDAC (15)
DNA Alkylation (13)
Amino Acids and Derivatives (13)
MRP (13)
Reverse Transcriptase (13)
Tyrosine Kinases (12)
TNF (12)
ATPase (11)
FLT (11)
FGFR (10)
DNA gyrase (10)
IL Receptor (10)
JAK (10)
Dopamine Receptor (10)
CDK (10)
Thrombin (10)
Retinoid Receptor (10)
Raf (10)
PKC (10)
Src (9)
Parasite (9)
DHFR (9)
c-Met/HGFR (9)
Lipoxygenase (9)
HIV Protease (8)
Endogenous Metabolite (8)
c-RET (8)
ALK (8)
NADPH (8)
NMDAR (7)
Proton pump (7)
ribosome (7)
ROS (7)
PI3K (7)
Aromatase (7)
HMG-CoA Reductase (7)
HIF (6)
ABC (6)
Phospholipase (6)
Proteasome (6)
STAT (6)
Serine Protease (6)
TAM Receptor (6)
TRP/TRPV Channel (6)
Tyrosinase (6)
PKA (5)
Prostaglandin Receptor (5)
mTOR (5)
MPO (5)
Antifungal (5)
CFTR (5)
CAT (5)
Hedgehog/Smoothened (5)
HER (5)
HSV (5)
Integrin (5)
MEK (5)
MMP (5)
HCV Protease (5)
HBV (5)
GluR (5)
GSK-3 (4)
DNA Methyltransferase (4)
Factor Xa (4)
Fatty Acid Synthase (4)
IκB/IKK (4)
Hydroxylase (4)
CaMK (4)
BCL (4)
BTK (4)
Antiviral (4)
Adenosine Receptor (4)
AMPK (4)
NOS (4)
PARP (4)
Opioid Receptor (4)
SGLT (4)
S1P Receptor (4)
Reductase (4)
UGT (4)
Transferase (4)
Trk receptor (4)
Thyroid hormone receptor(THR) (3)
Vasopressin Receptor (3)
Nucleoside Antimetabolite/Analog (3)
p38 MAPK (3)
Na-K-Cl cotransporter (3)
Annexin A (3)
AhR (3)
5-HT Receptor (3)
Arginase (3)
CXCR (3)
Cysteine Protease (3)
Chloride channel (3)
DPP-4 (3)
HSP (3)
LTR (3)
LDL (3)
GNRH Receptor (3)
GPCR19 (3)
GPR (3)
Free radical scavengers (3)
FXR (3)
Glucokinase (3)
Glutathione reductase (2)
GST (2)
Gap Junction Protein (2)
MAPK (2)
HIF/HIF Prolyl-Hydroxylase (2)
DNA (2)
Decarboxylase (2)
CCR (2)
Caspase (2)
CaSR (2)
Chk (2)
ATP Citrate Lyase (2)
ACAT (2)
AChE (2)
Akt (2)
Aminopeptidase (2)
Lipid (2)
Norepinephrine (2)
NOD (2)
P2 Receptor (2)
P-gp (2)
Phosphatase (2)
Rho (2)
ROCK (2)
ROR (2)
Sirtuin (2)
Serine/threonin kinase (2)
Syk (2)
Protease-activated Receptor (2)
PLK (2)
Wnt/beta-catenin (2)
TLR (2)
TGF-beta/Smad (2)
Telomerase (1)
VDA (1)
PKM (1)
Platelet aggregation (1)
RAR/RXR (1)
Ras (1)
Phosphorylase (1)
Somatostatin (1)
Serotonin Transporter (1)
Smo (1)
S6 Kinase (1)
PDK (1)
PED (1)
p53 (1)
PAFR (1)
OX Receptor (1)
NOD-like Receptor (NLR) (1)
NKCC (1)
NPC1L1 (1)
Nrf2 (1)
MT Receptor (1)
MTH1 (1)
Neurokinin receptor (1)
NADPH-oxidase (1)
ACK (1)
Acyltransferase (1)
advanced glycation end products (1)
ATM/ATR (1)
Aurora Kinase (1)
BACE (1)
Apoptosis (1)
Apoptosis inducer (1)
Antioxidant (1)
Antifolate (1)
Cell wall (1)
c-Fms (1)
Beta-Secretase (1)
cAMP (1)
Cannabinoid Receptor (1)
CSF-1R (1)
cholecystokinin (1)
DNA Alkylator/Crosslinker (1)
DUB (1)
Histone Demethylase (1)
Histone Methyltransferase (1)
Hexokinase (1)
Hydrogenase (1)
IAP (1)
IGF-1R (1)
Influenza Virus (1)
Integrase (1)
Mdm2 (1)
Melatonin Receptor (1)
Monoamine Transporter (1)
Monocarboxylate transporter (1)
Mitochondrial Metabolism (1)
Mitophagy (1)
Lipase (1)
lysosomal autophagy (1)
JNK (1)
GHSR (1)
GluCls (1)
Ferroptosis (1)
FAK (1)
Electron transport (1)
Endothelin Receptor (1)
Ephrin Receptor (1)
Epigenetic Reader Domain (1)
ERK (1)
Guanylate cyclase (1)
Hck (1)
GlyT (1)