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Compound Libraries Anti-cancer Active Compound library

Anti-cancer Active Compound library

Catalog No. L2160
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1656 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 18994.00
250 μL * 10 mM (in DMSO) 31171.00
1 mg 31171.00
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Product Description

  • A unique collection of 1656 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
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Library Composition

VEGFR (64)
PI3K (60)
EGFR (55)
CDK (52)
DNA/RNA Synthesis (45)
FGFR (41)
PDGFR (40)
Bcr-Abl (37)
c-Kit (36)
FLT (36)
mTOR (35)
c-Met/HGFR (34)
HDAC (33)
Topoisomerase (30)
Src (30)
JAK (27)
Microtubule Associated (27)
NF-κB (25)
Raf (25)
Estrogen/progestogen Receptor (24)
Apoptosis (23)
Akt (22)
HSP (22)
STAT (22)
ALK (21)
Autophagy (21)
MEK (20)
Epigenetic Reader Domain (20)
DNA-PK (19)
TNF (19)
PKC (19)
Tyrosine Kinases (18)
Dehydrogenase (17)
Aurora Kinase (17)
DNA Alkylation (16)
BCL (16)
TAM Receptor (16)
COX (15)
c-RET (15)
HER (15)
Endogenous Metabolite (14)
Androgen Receptor (13)
PARP (13)
P450 (12)
FAK (12)
ERK (12)
IGF-1R (12)
HIF (11)
ATM/ATR (11)
p38 MAPK (11)
Mdm2 (11)
PPAR (10)
Retinoid Receptor (10)
S6 Kinase (10)
Wnt/beta-catenin (10)
Caspase (10)
BTK (10)
IL Receptor (10)
Histone Methyltransferase (10)
Hedgehog/Smoothened (9)
Chk (9)
Trk receptor (9)
TGF-beta/Smad (9)
PLK (9)
Proteasome (9)
p53 (9)
Antioxidant (8)
Antiviral (8)
AChR (8)
GSK-3 (8)
HIV Protease (8)
GR (7)
MAO (7)
MMP (7)
IDO (7)
Histamine Receptor (7)
Glucocorticoid Receptor (7)
Adrenergic Receptor (7)
Antibacterial (7)
Calcium Channel (7)
CSF-1R (7)
CXCR (7)
c-Fms (6)
Antibiotic (6)
Apoptosis inducer (6)
Aromatase (6)
Gamma-secretase (6)
Histone Demethylase (6)
P-gp (6)
Pim (6)
Potassium Channel (6)
ROS (6)
TLR (6)
Vitamin (6)
Sodium Channel (5)
PDE (5)
Ras (5)
PKA (5)
PDK (5)
NOS (5)
GABA Receptor (5)
IκB/IKK (5)
Lipoxygenase (5)
IAP (5)
Integrin (5)
JNK (5)
Antifungal (5)
AMPK (5)
Adenosine Receptor (5)
CaMK (5)
Dopamine Receptor (5)
Cysteine Protease (4)
CCR (4)
Casein Kinase (4)
Antifection (4)
ATPase (4)
MAPK (4)
HBV (4)
Glucokinase (4)
DUB (4)
Phosphatase (4)
Phospholipase (4)
ROCK (4)
Serine Protease (4)
Sirtuin (4)
Transferase (4)
transporter (4)
UGT (3)
Tyrosinase (3)
Survivin (3)
Syk (3)
Tie-2 (3)
S1P Receptor (3)
Rho (3)
PYK2 (3)
Prostaglandin Receptor (3)
PAK (3)
Opioid Receptor (3)
NAMPT (3)
Monocarboxylate transporter (3)
E1/E2/E3 Enzyme (3)
Ephrin Receptor (3)
Fatty Acid Synthase (3)
GNRH Receptor (3)
Liver X Receptor (3)
LPA Receptor (3)
lysosomal autophagy (3)
Kinesin (3)
Annexin A (3)
Aminopeptidase (3)
5-HT Receptor (3)
cell cycle arrest (3)
Beta Amyloid (3)
DHFR (3)
cholecystokinin (3)
DNA Methyltransferase (3)
DNA Alkylator/Crosslinker (2)
Carbonic Anhydrase (2)
Chloride channel (2)
c-Myc (2)
AhR (2)
Amino Acids and Derivatives (2)
ATP Citrate Lyase (2)
BCRP (2)
KSP (2)
HSV (2)
Hydroxylase (2)
Mitophagy (2)
GPX (2)
GTPase (2)
Hexokinase (2)
MRP (2)
NADPH (2)
OXPHOS (2)
NMDAR (2)
NOD (2)
p97 (2)
Reactive Oxygen Species (2)
Reductase (2)
ROR (2)
TOPK (2)
STING (2)
Wee1 (2)
VDA (1)
TRP/TRPV Channel (1)
Xanthine Oxidase (1)
Smo (1)
Stemness kinase (1)
Thioredoxin (1)
Thrombin (1)
Telomerase (1)
ribosome (1)
Reverse Transcriptase (1)
Serine/threonin kinase (1)
Serotonin Transporter (1)
SGK (1)
SGLT (1)
Sigma receptor (1)
SIK (1)
RAAS (1)
PTEN (1)
Protease-activated Receptor (1)
Porcupine (1)
PKM (1)
PAFR (1)
Parasite (1)
PD-1/PD-L1 (1)
PI4K (1)
Nrf2 (1)
Nucleoside Antimetabolite/Analog (1)
MTH1 (1)
MPO (1)
HIF/HIF Prolyl-Hydroxylase (1)
Hck (1)
HCV Protease (1)
GPCR19 (1)
GPR (1)
Ferroptosis (1)
GluR (1)
GHSR (1)
Estrogen Receptor/ERR (1)
Free radical scavengers (1)
MNK (1)
Melatonin Receptor (1)
MELK (1)
MALT (1)
LTR (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Influenza Virus (1)
LHRH (1)
Lipase (1)
IRAK (1)
Isocitrate Dehydrogenase (IDH) (1)
ASK (1)
Antifolate (1)
Adiponectin receptor (1)
ABC (1)
AChE (1)
ACK (1)
DPP-4 (1)
Discoidin Domain Receptor (DDR) (1)
Dehydrogenase inhibitor (1)
Deubiquitinase (1)
CRM1 (1)