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WZ4002  
Catalog No. T6238    CAS 1213269-23-8
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Availability
Price/USD
Quantity
5mg
In stock
40.00
10mg
In stock
60.00
25mg
In stock
101.00
50mg
In stock
170.00
100mg
In stock
298.00
1g
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0.00
5g
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0.00
10 mM * 1 mL (in DMSO)
In stock
65.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.12% COA Datasheet HNMR HPLC
Biological Activity:

Product Description:

WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 nM.

Target:
EGFR (L858R/T790M); EGFR (L858R);
Research Area:
Cancer
Chemical Information:
Molecular Weight 494.18
Formula C25H27ClN6O3
CAS Number 1213269-23-8
Solubility DMSO:11 mg/mL (22.3 mM);Ethanol:<1 mg/mL;Water:<1 mg/mL
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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