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Home > Immunology/Inflammation > TGF/beta/Smad > LY2109761
LY2109761  
Catalog No. T2123    CAS 700874-71-1
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2mg
In stock
40.00
5mg
In stock
77.00
10mg
In stock
128.00
25mg
In stock
218.00
50mg
In stock
383.00
100mg
In stock
587.00
200mg
In stock
842.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
84.00
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Documents and Quality Management
Purity:99.83% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

LY2109761 is a novel selective TGF-β receptor type I/II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM, respectively; shown to negatively affect the phosphorylation of Smad2.

Target:
TGF-β receptor typeII; TGF-β receptor type I;
Research Area:
Immunology
Chemical Information:
Molecular Weight 441.52
Formula C26H27N5O2
CAS Number 700874-71-1
Solubility DMSO: 2mg/ml(4.53 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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