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Home > Tyrosine Kinase/Adaptors > IGF/1R > GSK1838705A
GSK1838705A  
Catalog No. T3079    CAS 1116235-97-2
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2mg
In stock
67.00
5mg
In stock
128.00
10mg
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213.00
25mg
In stock
362.00
50mg
In stock
638.00
100mg
In stock
808.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
150.00
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Documents and Quality Management
Purity:98.89% COA Datasheet HNMR LCMS MSDS
Biological Activity:

Product Description:

GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein kinases.

Target:
RSK1; insulin receptor; IGF-1R; ALK;
Research Area:
Cancer
Chemical Information:
Molecular Weight 532.57
Formula C27H29FN8O3
CAS Number 1116235-97-2
Solubility DMSO: 107mg/ml(200.91 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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