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Enasidenib  
Catalog No. T2346    CAS 1446502-11-9
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5mg
In stock
60.00
10mg
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85.00
25mg
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143.00
50mg
In stock
247.00
100mg
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417.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
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65.00
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Documents and Quality Management
Purity:99.45% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

Enasidenib is an orally available inhibitor of specific mutant forms of the mitochondrial enzyme isocitrate dehydrogenase type 2 (IDH2), with potential antineoplastic activity.

Target:
IDH2;
Research Area:
Other
Chemical Information:
Molecular Weight 473.38
Formula C19H17F6N7O
CAS Number 1446502-11-9
Solubility DMSO:10 mM;Ethanol:100 mg/mL (211.25 mM);Water:<1 mg/mL
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Product Recommendations
  • AGI-5198 (IDH-C35), AGI-5198 is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μ...
  • IDH1-IN-1, Mutant IDH1-IN-1 is a potent mutant IDH1 R132 h inhibitor with IC50 < 0.1 uM.
  • AGI-6780, AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.

 

Reference

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