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Home > Immunology/Inflammation > HDAC > Droxinostat
Droxinostat  
Catalog No. T6481    CAS 99873-43-5
Pack Size
Availability
Price/USD
Quantity
10mg
9 days
67.00
10mM * 1mL (in DMSO)
9 days
57.00
100mg
9 days
518.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

Droxinostat is a selective inhibitor of HDAC, mostly for HDACs 6 and 8 with IC50 of 2.47 μM and 1.46 μM, greater than 8-fold selective against HDAC3 and no inhibition to HDAC1, 2, 4, 5, 7, 9, and 10.

Target:
HDAC10; HDAC9 ; HDAC3 ; HDAC6 ; HDAC8 ;
Research Area:
Cancer
Chemical Information:
Molecular Weight 243.69
Formula C11H14ClNO3
CAS Number 99873-43-5
Solubility DMSO: 49mg/ml(201.08 mM);Water: <1mg/ml;Ethanol: 49mg/ml(201.08 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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