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Cilomilast  
Catalog No. T6445    CAS 153259-65-5
Pack Size
Availability
Price/USD
Quantity
5mg
9 days
71.00
10mM * 1mL (in DMSO)
9 days
94.00
100mg
9 days
518.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

Cilomilast is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.

Target:
LPDE4; HPDE4;
Research Area:
Metabolism system
Chemical Information:
Molecular Weight 343.42
Formula C20H25NO4
CAS Number 153259-65-5
Solubility DMSO:69 mg/mL (200.92 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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