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Home > Cell cycle/Check point > HDAC > CUDC-101
CUDC-101  
Catalog No. T3108    CAS 1012054-59-9
Pack Size
Availability
Price/USD
Quantity
2mg
In Stock
44.00
25mg
In Stock
193.00
50mg
In Stock
309.00
100mg
In Stock
459.00
10mM * 1mL (in DMSO)
In Stock
83.00
10mg
In Stock
74.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:96.26% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

CUDC-101 is a potent multi-targeted inhibitor against HDAC, EGFR and HER2 with IC50 of 4.4 nM, 2.4 nM, and 15.7 nM, and inhibits class I/II HDACs, but not class III, Sir-type HDACs. Phase 1.

Target:
EGFR; HDACs;
Research Area:
Cancer
Chemical Information:
Molecular Weight 434.49
Formula C24H26N4O4
CAS Number 1012054-59-9
Solubility DMSO: 20mg/ml(46.03 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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