||BX-517 is a potent and selective inhibitor of PDK1.
||Dichloroacetate ion inhibits pyruvate dehydrogenase kinase, resulting in the inhibiti...
||AR-12 is an orally bioavailable, small-molecule, celecoxib-derived inhibitor of phosp...
||PHT-427 is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity bi...
||GSK2334470 is a novel PDK1 inhibitor (IC50: ~10 nM, in a cell-free assay), with no in...
||BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: ...
||BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity ...