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Metabolism-Others
Cat.No. Product Name Information Area
T4415 Katacine Katacine inhibits of oxygen consumption and suppresses the speed of electrons transfe... Respiration and Oxidation
T4410 LM10 Selective tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50 values are 0.62 and 2 μM f... Metabolic disease
T4379 Tropifexor Tropifexor is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM. digestive disease(hepatobiliary disease)
T4359 VAS2870 VAS2870 is a NADPH oxidase (NOX) inhibitor. Cardiovascular diseases
T4354 KPT-9274 KPT-9274 is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is ... Cancer
T6301 Tosedostat (CHR2797) CHR-2797 is an orally bioavailable inhibitor of the M1 family of aminopeptidases with... Cancer
T4335 GNE-617 GNE-617, a specific NAMPT inhibitor(IC50=5 nM), shows potency in xenograft models of ...
T4308 F1063-0967 F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11... others
T4280 LTI-291 LTI-291 is a glucocerebrosidase (Gcase) activator. Nervous system disease
T4253 Skp2 Inhibitor C1 Skp2 Inhibitor C1(SKPin C1) is a specific small molecule inhibitor of Skp2-mediated p... others
T4254 TM5441 TM5441 is an orally bioavailable inhibitor of plasminogen activator inhibitor 1 (PAI-...
T4255 TM5275 sodium TM5275 is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).
T4256 PTP1B-IN-2 PTP1B-IN-2 is an effective protein tyrosine phosphatase 1B (PTP1B) inhibitor(IC50=50 ... others
T4277 Osilodrostat Osilodrostat (LCI699) is an effective inhibitor of human 11β-hydroxylase (IC50: 2.5 n... Endocrine
T4200 AHU377 AHU-377 hemicalcium salt is a potent NEP inhibitor with an IC50 of 5 nM. AHU-377 is a... Others
T4170 PKM2 inhibitor PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of ... Others
T4192 hnps-PLA Inhibitor Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (... Others
T4188 SDZ285-428 NVP-VID-400 (SDZ285-428) is a CYP24A1 inhibitor. Others
T4179 Probucol disuccinate Probucol is an anti-hyperlipidemic drug initially developed in the treatment of coron... Others
T4467 UAMC 00039 dihydrochloride UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidas... Others
T4114 Diffractaic Acid Diffractaic Acid can inhibit LTB4 biosynthesis in A-23187-stimulated bovine PMNL cell... Others
T4052 KML29 KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor. It ... Others
T4050 GSK2981278 GSK2981278 is a highly potent and selective inverse agonist of retinoic acid receptor... Immunology
T4039 BIBB 515 BIBB 515 is a selective and potent inhibitor of OSC in vivo with an ED50 value of 0.2... Others
T3976 Cytosporone B Cytosporone B is a naturally occurring agonist for the nuclear receptor Nur77 (IC50 =... Others
T3529 Bestatin hydrochloride Bestatin (Ubenimex) hydrochlorideis an inhibitor of aminopeptidase N (APN)/CD13 and a... Others
T3580 FIPI FIPI is a derivative of halopemide which potently inhibits both PLD1 (IC50 = 25 nM) a... Others
T3970 XL-652 BMS-779788 is an LXRα/β partial agonist (IC50: 68/14 nM). cardiovascular system
T3585 TMS TMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). Cancer
T3797 Isosilybin Isosilybin and Silybin might be suitable candidates to design potent PXR antagonists ... Others
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