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Metabolism-Others
Cat.No. Product Name Information Area
T4379 Tropifexor Tropifexor is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM. digestive disease(hepatobiliary disease)
T4359 VAS2870 VAS2870 is a NADPH oxidase (NOX) inhibitor. Cardiovascular diseases
T4354 KPT-9274 KPT-9274 is an orally bioavailable small molecule that is a non-competitive dual inhi... Cancer
T6301 Tosedostat (CHR2797) Cancer
T4335 GNE-617 GNE-617 is a specific NAMPT inhibitor that inhibits the biochemical activity of NAMPT...
T4308 F1063-0967 F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11... others
T4280 LTI-291 LTI-291 is an activator of glucocerebrosidase (Gcase) extracted from patent WO 201719... Nervous system disease
T4253 Skp2 Inhibitor C1 Skp2 Inhibitor C1(SKPin C1) is a specific small molecule inhibitor of Skp2-mediated p... others
T4254 TM5441 TM5441 is an orally bioavailable inhibitor of plasminogen activator inhibitor 1 (PAI-... others
T4255 TM5275 sodium TM5275 is an inhibitor of plasminogen activator inhibitor 1 (PAI-1; IC50 = 6.95 ?M), ... others
T4256 PTP1B-IN-2 PTP1B-IN-2 is a potent protein tyrosine phosphatase 1B (PTP1B) inhibitor with an IC50... others
T4277 Osilodrostat Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase and aldosterone ... Endocrine
T4200 AHU377 AHU-377 hemicalcium salt is a potent NEP inhibitor with an IC50 of 5 nM. AHU-377 is a... Others
T4170 PKM2 inhibitor PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of ... Others
T4192 hnps-PLA Inhibitor Hnps-PLA Inhibitor, is an inhibitor of human nonpancreatic secretory Phospholipase A ... Others
T4188 SDZ285-428 NVP-VID-400, also known as SDZ285-428, is CYP24A1 inhibitor. Others
T4179 Probucol disuccinate Probucol is an anti-hyperlipidemic drug initially developed in the treatment of coron... Others
T4467 UAMC 00039 dihydrochloride UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidas... Others
T4114 Diffractaic Acid Inhibition of LTB4 biosynthesis in A-23187-stimulated bovine PMNL cells with activity... Others
T4052 KML29 Highly selective and potent monoacylglycerol lipase (MAGL) inhibitor. Exhibits potent... Others
T4050 GSK2981278

GSK2981278 is a highly potent and selective inverse agonist of retinoic acid recep...

Immunology
T4039 BIBB 515 BIBB 515 is a selective and potent inhibitor of OSC in vivo with an ED50 value of 0.2... Others
T3976 Cytosporone B ytosporone B is a naturally occurring agonist for the nuclear receptor Nur77 (IC50 = ... Others
T3529 Bestatin hydrochloride Bestatin (Ubenimex) hydrochlorideis an inhibitor of aminopeptidase N (APN)/CD13 and a... Others
T3580 FIPI FIPI is a derivative of halopemide which potently inhibits both PLD1 (IC50 = 25 nM) a... Others
T3970 XL-652 BMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for ... cardiovascular system
T3585 TMS TMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). It has... Cancer
T3797 Isosilybin Isosilybin and Silybin might be suitable candidates to design potent PXR antagonists ... Others
T3763 Fumaric acid Fumaric acid is used in systemic and topical treatment of psoriasis. Fumaric acid att... Others
T3756 Allitol Allitol is useful as a sweetener and the raw material for production of chemical comp... Others
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