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Metabolism-Others
Cat.No. Product Name Information Area
T4052 KML29 Highly selective and potent monoacylglycerol lipase (MAGL) inhibitor. Exhibits potent... Others
T4050 ROR gama modulator 1 GSK2981278 is a highly potent and selective inverse agonist of retinoic acid receptor... Immunology
T4039 BIBB 515 BIBB 515 is a selective and potent inhibitor of OSC in vivo with an ED50 value of 0.2... Others
T3976 Cytosporone B ytosporone B is a naturally occurring agonist for the nuclear receptor Nur77 (IC50 = ... Others
T3529 Bestatin hydrochloride Bestatin (Ubenimex) hydrochlorideis an inhibitor of aminopeptidase N (APN)/CD13 and a... Others
T3580 FIPI FIPI is a derivative of halopemide which potently inhibits both PLD1 (IC50 = 25 nM) a... Others
T3970 XL-652 BMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for ... cardiovascular system
T3585 TMS TMS is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1). It has... Cancer
T3797 Isosilybin Isosilybin and Silybin might be suitable candidates to design potent PXR antagonists ... Others
T3763 Fumaric acid Fumaric acid is used in systemic and topical treatment of psoriasis. Fumaric acid att... Others
T3756 Allitol Allitol is useful as a sweetener and the raw material for production of chemical comp... Others
T3420 CA-074 methyl ester CA-074 methyl ester is a specific inhibitor of Cathepsin B, which has potent bioactiv... Other
T3715 Acebilustat Acebilustat, also known as ZK322, is a potent and selective leukotriene B4 hydrolase ... Metabolism
T3666 Atractylodin Atractylodin has high lipase inhibitory activity (IC50?=?39.12?μM); Atractylodin poss... Others
T3669 Curcumenol Curcumenol, one of the major components of Zedoary turmeric oil, is an antibiotic dru... Others
T6893 MK-886 (L-663,536) MK-886 is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activat... Others
T6800 CCF642 CCF642 is a novel PDI-inhibiting compound with antimyeloma activity. Others
T6795 Carbidopa Carbidopa is an aromatic-L-amino-acid decarboxylase inhibitor with an IC50 of 29 ± 2 ... Others
T3428 Helicidnew Helicid is a medicine available in a number of countries worldwide. Others
T3418 demethylzeylasteralnew Demethylzeylasteral has strong immunosuppressive activity, can be used in the fields ... Cancer/ Immunology
T3617 Ivosidenibnew Ivosidenib is an orally available inhibitor of isocitrate dehydrogenase type 1 (IDH1)... Cancer
T0140 Sibutramine Sibutramine (trade name Meridia in the USA, Reductil in Europe and Others countries),... Metabolism system
T3315 Benurestat Benurestat, a urease inhibitor for the therapy of infected ureolysis. Other
T3268 Mildronate Mildronate is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB... Cardiovascular System
T2172 SQ 22536 The adenosine analogue 9-(Tetrahydro-2-furyl)adenine, SQ 22536, inhibited adenylate c... Others
T6625 Ozagrel hydrochloride Ozagrel HCl is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC5... Metabolism system
T6690 T0901317 T0901317 is a potent and selective agonist for both LXR and FXR, with EC50 of ~50 nM ... Metabolism system
T2545 Lomitapide Mesylate Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibi... Metabolism system
T3104 LY2608204 LY2608204 activates glucokinase (GK) with EC50 of 42 nM. Phase 2. Metabolism system
T2968 Hyodeoxycholic acid (HDCA) Extracted from Pigs bile;Suitability:alcohol;Store the product in sealed,cool and dry... Metabolism system
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