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GPCR-G Protein-Others
Cat.No. Product Name Information Area
T3520 Setipiprant Setipiprant is an orally available, selective CRTH2 antagonist. CRTH2 is a G protein-... Others
T4016 BMS-986020 BMS-986020 is an LPA1 antagonist. target: LPA1 BMS-986020 is in Phase 2 clinical deve... Others
T3993 BQCA BQCA a highly selective allosteric modulator of the M1 mAChR. Others
T3967 Exendin-4 Exendin-4, a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor... Others
T3965 Fevipiprant Fevipiprant(QAW039) is a selective, potent, reversible competitive CRTh2 antagonist w... Others
T3565 UV0155041 UV0155041 is a potent, positive allosteric modulator/allosteric agonist at mGlu4 rece... Others
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and... Other
T3148 MK571 MK-571 is a selective, orally active?CysLT1 receptor(Cysteinyl leukotriene receptor)?... Respiratory?system/ Cardiovascular system
T3630 Relugolix Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH... Cancer/ Nervous system
T7013 Vorapaxar

Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) ant...

T3597 Cutamesine dihydrochloridenew Selective?σ1 receptor agonist (IC50?= 17.4 nM). Exhibits selectivity for?σ1 over?σ2 r... Immunology
T3258 Ponesimod Ponesimod(ACT-128800) is an orally active, selective sphingosine-1-phosphate receptor... Immunology
T3216 Selexipag(NS-304) NS-304 is an orally available and potent agonist for the PGI(2) receptor (IP receptor... Other
T3177 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist is a potent (EC50 on OX2R is 23 nM) and OX2R-selective (OX1... Other
T3185 R112 R112 is an ATP-competitive inhibitor of Syk kinase with a Ki of 96 nM. R112 inhibits ... Immunology
T3174 Taprenepag Taprenepag (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (E... Immunology
T3194 Ro 46-2005 Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits ... Cardiovascular System
T3178 BIBS 39 BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist. Cardiovascular System
T3040 Gallein Gallein is a small molecule inhibitor of Gβγ activity. Cardiovascular System
T6590 MK-3207 hydrochloride MK-3207 is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM,... Nervous system
T6108 Ki16425 Ki16425 is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 wit... Cancer
T2126 MK5046 MK-5046 is a novel BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 n... Other
T2086 ELN 441958 ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of th... Other
T2000 AM095 AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 _mu_M fo... Other
T1978 GW627368 GW627368(GW627368X) is a novel, potent and selective competitive antagonist of prosta... Other
T1824 TGR5 Receptor Agonist TGR5 Receptor Agonist, a potent TGR5(GPCR19) agonist, showed improved potency in the ... Other
T1677L Montelukast sodium Montelukast sodium is a leukotriene receptor antagonist (LTRA) used for the maintenan... Cancer
T1626 Prostaglandin E1 Prostaglandin E1 (Alprostadil) is a prostaglandin, which is used in the treatment of ... Cardiovascular System