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Home > GPCR-G Protein-Others
GPCR-G Protein-Others
Cat.No. Product Name Information Area
T4546 Dinoprost Tromethamine Dinoprost(Prostaglandin F2α) tromethamine salt is a naturally occurring prostaglandin... Others
T4648 TC-G-1008 TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat ... Metabolic Disease
T4390 ML221 ML221 is a potent?apelin /APJ?functional antagonist, inhibiting apelin-13-mediated ac...
T1418 Bucladesine sodium salt Bucladesine, PKA activator, is a cyclic nucleotide derivative that mimics the action ... anti-infection
T4278 AM966 AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses L... cancer
T4300 AZD2098 AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research... Inflammation
T7040 Angiotensin II human Angiotensin II is mediated by AT1 and AT2 receptors. AT1 and AT2 receptors have seven... cancer
T4186 AC-264613 AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 s... Others
T4540 ML 18 ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of... Others
T4500 ADX88178 ADX88178 is a potent positive allosteric modulator for metabotropic glutamate recepto... Others
T4352 SB-756050 SB756050 is a specific TGR5 agonist. Others
T4119 Octreotide Acetate Octreotide acetate is a potent, long-acting synthetic somatostatin octapeptide analog... Metbolism/ Cancer
T4102 Goserelin acetate Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormon... Cancer
T4083 BAR 501 BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM). Other
T3520 Setipiprant Setipiprant is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 ... Others
T4016 BMS-986020 BMS-986020 is a selective antagonist of LPA1. Others
T3993 BQCA BQCA a highly selective allosteric modulator of the M1 mAChR. Others
T3967 Exendin-4 Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exen... Others
T3965 Fevipiprant Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist. Others
T3565 UV0155041 UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGl... Others
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor. Other
T3148 MK571 MK-571 is a selective, orally active?antagonist of the CysLT1 receptor. MK571 is a mu... Respiratory system/ Cardiovascular system
T3630 Relugolix Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or... Cancer/ Nervous system
T7013 Vorapaxar Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) an... Others
T3597 Cutamesine dihydrochloridenew Cutamesine dihydrochloride is a selective?σ1 receptor agonist (IC50: 17.4 nM). It sho...
T3258 Ponesimod Ponesimod is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) ago... Immunology
T3216 Selexipag(NS-304) Selexipag(NS-304) is prostacyclin receptor agonist that causes vasodilation in pulmon... Other
T3177 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R... Other
T3185 R112 R112 is an ATP-competitive inhibitor of Syk kinase. Immunology
T3174 Taprenepag Taprenepag (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (E... Immunology
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