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GPCR-G Protein-Others
Cat.No. Product Name Information Area
T4390 ML221

ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated...

T1418 Bucladesine sodium salt Bucladesine is a cell-permeable PKA activator by mimicing the action of endogenous cA... anti-infection
T4278 AM966 AM966 is a high affinity, selective, oral LPA1-antagonist, inhibits LPA-stimulated in... cancer
T4300 AZD2098 AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor, used for asthma researc... Inflammation
T7040 Angiotensin II human Angiotensin II human is converted by Angiotensin I through removal of two C-terminal ... cancer
T4186 AC-264613 AC-264613 is the first agonist of the G-protein-coupled receptor (GPCR) protease acti... Others
T4540 ML 18 ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of... Others
T4500 ADX88178 DX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor... Others
T4352 SB-756050 SB756050 is a selective TGR5 agonist currently in phase 1clinical trials for the trea... Others
T4119 Octreotide acetate Octreotide (acetate) is a long-acting octapeptide and somatostatin analog with pharma... Metbolism/ Cancer
T4102 Goserelin acetate

Goserelin (ICI 118630) acetate is an injectable gonadotropin releasing hormone sup...

Cancer
T4083 BAR 501 BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM. Other
T3520 Setipiprant Setipiprant is an orally available, selective CRTH2 antagonist. CRTH2 is a G protein-... Others
T4016 BMS-986020 BMS-986020 is an LPA1 antagonist. target: LPA1 BMS-986020 is in Phase 2 clinical deve... Others
T3993 BQCA BQCA a highly selective allosteric modulator of the M1 mAChR. Others
T3967 Exendin-4 Exendin-4, a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor... Others
T3965 Fevipiprant Fevipiprant(QAW039) is a selective, potent, reversible competitive CRTh2 antagonist w... Others
T3565 UV0155041 UV0155041 is a potent, positive allosteric modulator/allosteric agonist at mGlu4 rece... Others
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and... Other
T3148 MK571 MK-571 is a selective, orally active?CysLT1 receptor(Cysteinyl leukotriene receptor)?... Respiratory?system/ Cardiovascular system
T3630 Relugolix Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH... Cancer/ Nervous system
T7013 Vorapaxar Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antago... Others
T3597 Cutamesine dihydrochloridenew Selective?σ1 receptor agonist (IC50?= 17.4 nM). Exhibits selectivity for?σ1 over?σ2 r... Immunology
T3258 Ponesimod Ponesimod(ACT-128800) is an orally active, selective sphingosine-1-phosphate receptor... Immunology
T3216 Selexipag(NS-304) NS-304 is an orally available and potent agonist for the PGI(2) receptor (IP receptor... Other
T3177 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist is a potent (EC50 on OX2R is 23 nM) and OX2R-selective (OX1... Other
T3185 R112 R112 is an ATP-competitive inhibitor of Syk kinase with a Ki of 96 nM. R112 inhibits ... Immunology
T3174 Taprenepag Taprenepag (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (E... Immunology
T3194 Ro 46-2005 Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits ... Cardiovascular System
T3178 BIBS 39 BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist. Cardiovascular System
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