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Epigenetic-Reader-Domain
Cat.No. Product Name Information Area
T6389 Anacardic Acid Anacardic Acid is a potent inhibitor of p300 and p300/CBP-associated factor histone a... Cancer
T4345 CeMMEC1 CeMMEC1 is an inhibitor of BRD4, and also has high affinity for TAF1, with an IC50 of...
T3504 AZD5153 AZD 5153 an orally available, bivalent inhibitor of the bromodomain and extraterminal... Others
T3712 Mivebresib Mivebresib, also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-cont... Cancer
T3311 GSK6853 GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhi... Others
T6939 PFI-3 PFI-3 is a selective chemical probe for SMARCA bromodomains, including SMARCA2, SMARC... Others
T6859 I-BRD9 I-BRD9 is the first selective cellular chemical probe for BRD9 (pIC50=7.3). others
T6811 CPI-637 CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibit... Others
T6786 BI-9564 BI-9564 is a selective, and cell-permeable BRD9 BD inhibitor, with Kd of 5.9 nM for B... others
T6783 BI-7273 BI-7273 is a potent, selective, and cell-permeable BRD9 BD Inhibitor. Others
T6668 SGC-CBP30 SGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50 of 21 nM and 38 nM, respective... Cancer
T6255 Bromosporine Bromosporine is a broad spectrum inhibitor for bromodomains with IC50 of 0.41 μM, 0.2... others
T6222 PFI-1 (PF-6405761) PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC5... Cancer
T6032 OTX015 OTX015 is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for B... Cancer
T6021 GSK1324726A (I-BET726) GSK1324726A (I-BET726) is a highly selective inhibitor of BET family proteins with IC... Cancer
T2480 RVX-208 RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell... Cancer
T2436 GSK2801 GSK2801 is a potent, selective and cell active acetyl-lysine competitive inhibitor of... Cancer
T2379 UNC1215 UNC1215 is a potent and selective MBT (malignant brain tumor) antagonist, which binds... Cancer
T2252 UNC 669 UNC669 is a potent and selective MBT (malignant brain tumor) inhibitor with IC50 of 6... Other
T2110 (+)-JQ-1 (+)-JQ1 is a BET bromodomain inhibitor, with IC50 of 77 nM/33 nM for BRD4(1/2) in cel... Other
T2091 CPI-0610 CPI-0610 is a potent, selective, and cell-active BET bromodomain inhibitor CPI-0610 i... Other
T2072 BET bromodomain inhibitor It is a BET bromodomain inhibitor Other
T1906 GSK-525762A(I-BET-762) GSK 525762A (I-BET 762) is an inhibitor for BET proteins with IC50 of ~35 nM. Immunology
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