||MG149 is a potent histone acetyltransferase inhibitor with IC50 of 74 μM and 47 μM for Tip60 and MOF...
||INCB-28060(free base) is a novel, ATP-competitive inhibitor of c-MET kinase with an IC50 with 0.13 n...
||PF-06840003 is a highly selective orally bioavailable IDO-1 inhibitor.
||AM966 is a high affinity, selective, oral LPA1-antagonist, inhibits LPA-stimulated intracellular cal...
||THZ531 is a covalent inhibitor of both CDK12 and CDK13 with IC50s of 158 nM and 69 nM, respectively.
||LY2606368 is a potent and selective ATP competitive inhibitor of the Chk1 protein kinase, with IC50s...
||Ki-20227 is a highly selective c-Fms tyrosine kinase(CSF1R) inhibitor with IC50 value of 2 nM; 6 fol...
||Belizatinib is an oral, dual, potent inhibitor of ALK and TRKA, TRKB, and TRKC, with IC50 of 0.7?nM ...