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BRD4 Inhibitor-27

Name: BRD4 Inhibitor-27
Brand: TargetMol
SKU: T78555
Price: 82 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T78555Cas No. 930039-92-2

BRD4 Inhibitor-27 is a potent BRD4 inhibitor that inhibits BRD4 BD1 and BRD4 BD2 with IC50s of 9.6 and 11.3 μM, respectively.BRD4 Inhibitor-27 has anticancer activity and can be used for breast cancer research.

BRD4 Inhibitor-27

🥰Excellent

Purity: 99.22%

Catalog No. T78555Cas No. 930039-92-2

Pack Size	Price	Availability
1 mg	$82	In Stock
5 mg	$203	In Stock
10 mg	$291	In Stock
25 mg	$453	In Stock
50 mg	$625	In Stock
100 mg	$826	In Stock
200 mg	$1,110	In Stock

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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.22%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	BRD4 Inhibitor-27 is a potent BRD4 inhibitor that inhibits BRD4 BD1 and BRD4 BD2 with IC50s of 9.6 and 11.3 μM, respectively.BRD4 Inhibitor-27 has anticancer activity and can be used for breast cancer research.
Targets&IC50	BD1:9.6 uM, BD2:11.3 uM

Chemical Properties

Molecular Weight	346.31
Formula	C₁₆H₁₃F₃N₆
Cas No.	930039-92-2
Smiles	FC(F)(F)C1=NN=C2C=CC(NCCC3=CNC4=C3C=CC=C4)=NN12

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 55 mg/mL (158.82 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.8876 mL	14.4379 mL	28.8759 mL	144.3793 mL
5 mM	0.5775 mL	2.8876 mL	5.7752 mL	28.8759 mL
10 mM	0.2888 mL	1.4438 mL	2.8876 mL	14.4379 mL
20 mM	0.1444 mL	0.7219 mL	1.4438 mL	7.2190 mL
50 mM	0.0578 mL	0.2888 mL	0.5775 mL	2.8876 mL
100 mM	0.0289 mL	0.1444 mL	0.2888 mL	1.4438 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc